31 products were found matching "K22599"!
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Lopinavir
Item number: TGM-T1623-100mg
Description: Lopinavir (ABT-378) is a peptidomimetic HIV protease inhibitor effective against HIV protease with the Val 82 mutation. It is less affected by serum protein binding compared to the structurally related drug ritonavir. Target: SARS-CoV, HIV Protease. Smiles:...
| Keywords: | ABT-378 |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 192725-17-0 |
| MW: | 628.8 D |
From 42.00€
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Ritonavir
Item number: TGM-T1525-100mg
Description: Ritonavir (ABT 538) is a peptidomimetic agent that inhibits both HIV-1 and HIV-2 proteases. Ritonavir is highly inhibited by serum proteins but boosts the effect of other HIV proteases by blocking their degradation by cytochrome P450. Target: SARS-CoV, Apoptosis, HIV Protease. Smiles:...
| Keywords: | A 84538, ABT 538, RTV, Abbott 84538 |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 155213-67-5 |
| MW: | 720.94 D |
From 31.00€
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Brecanavir
Item number: TGM-T30585-100mg
Description: Brecanavir is a tyrosyl-based arylsulfonamide, high affinity, protease inhibitor (PI) for the treatment of human immunodeficiency virus type 1. Target: Others. Smiles: O(C(N[C@@H](CC1=CC=C(OCC=2N=C(C)SC2)C=C1)[C@@H](CN(S(=O)(=O)C=3C=C4C(=CC3)OCO4)CC(C)C)O)=O)[C@@H]5[C@]6([C@@](OC5)(OCC6)[H])[H]....
| Keywords: | CHEMBL206031, UNII-E367I8C7FI, GW-640385X, GW-0385, GW-640385 |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 313682-08-5 |
| MW: | 703.82 D |
From 1,671.00€
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Darunavir Ethanolate
Item number: TGM-T3335-100mg
Description: Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS. Due to the emergence of ANTIVIRAL DRUG RESISTANCE when used alone, it is administered in combination with other ANTI-HIV AGENTS. Target: HIV Protease. Smiles:...
| Keywords: | TMC114, Darunavir Ethanolate, UIC 94017 |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 635728-49-3 |
| MW: | 593.74 D |
From 31.00€
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Palinavir
Item number: TGM-T28292-100mg
Description: Palinavir is an antiviral, it inhibits HIV-1 protease. Target: Others. Smiles: C([C@H]([C@H](CC1=CC=CC=C1)NC([C@@H](NC(=O)C2=NC3=C(C=C2)C=CC=C3)[C@H](C)C)=O)O)N4[C@H](C(NC(C)(C)C)=O)C[C@H](OCC=5C=CN=CC5)CC4. References: Lamarre D, Croteau G, Wardrop E, Bourgon L, Thibeault D, Clouette C, Vaillancourt M,...
| Keywords: | BILA 2011 BS |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 154612-39-2 |
| MW: | 708.89 D |
From 1,971.00€
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Tipranavir
Item number: TGM-T4578-100mg
Description: Tipranavir is a protease inhibitor that inhibits HIV-1 resistant to more than 1 protease inhibitor .Tipranavir effectively inhibits HIV-1 protease enzyme activity and dimerisation and has potent activity against multiple protease inhibitor (PI) HIV-1 isolates (IC50 of 66-410 nM). Tipranavir inhibits...
| Keywords: | PNU-140690 |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 174484-41-4 |
| MW: | 602.66 D |
From 125.00€
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Indinavir sulfate
Item number: TGM-T5863-100mg
Description: Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM. Target: SARS-CoV, HIV Protease. Smiles: OS(O)(=O)=O.CC(C)(C)NC(=O)[C@@H]1CN(Cc2cccnc2)CCN1C[C@@H](O)C[C@@H](Cc1ccccc1)C(=O)N[C@@H]1[C@H](O)Cc2ccccc12....
| Keywords: | MK-639 sulfate, L735524 sulfate |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 157810-81-6 |
| MW: | 711.87 D |
From 58.00€
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Nelfinavir Mesylate
Item number: TGM-T6001-100mg
Description: Nelfinavir Mesylate (Viracept) is an effective HIV protease inhibitor (Ki: 2 nM). Target: HIV Protease. Smiles: Cc1c(cccc1O)C(=O)N[C@@H](CSc1ccccc1)[C@@H](CN1C[C@H]2CCCC[C@H]2C[C@H]1C(=O)NC(C)(C)C)O.CS(=O)(=O)O. References: Xiang T, et al. Y Lett. 2015 Aug 1,364(1):79-88.
| Keywords: | Nelfin, Viracept, AG1343, AG 1343 Mesylate |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 159989-65-8 |
| MW: | 663.89 D |
From 48.00€
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Fosamprenavir sodium
Item number: TGM-T69713-100mg
Description: Fosamprenavir sodium is an HIV protease inhibitor that is the water soluble prodrug of amprenavir. Target: Others. Smiles: [Na+].[Na+].CC(C)CN(C[C@@H](OP([O-])([O-])=O)[C@H](Cc1ccccc1)NC(=O)O[C@H]1CCOC1)S(=O)(=O)c1ccc(N)cc1
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 226700-80-7 |
| MW: | 629.57 D |
From 1,520.00€
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Indinavir monohydrate
Item number: TGM-T70166-100mg
Description: Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability. Target: Others. Smiles: O.CC(C)(C)NC(=O)[C@@H]1CN(Cc2cccnc2)CCN1C[C@@H](O)C[C@@H](Cc1ccccc1)C(=O)N[C@@H]1[C@H](O)Cc2ccccc12
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 180683-37-8 |
| MW: | 631.82 D |
From 2,272.00€
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Saquinavir
Item number: TGM-T7903-10mg
Description: Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS. Target: SARS-CoV, HIV Protease. Smiles: CC(C)(C)NC(=O)C1CC2CCCCC2CN1CC(O)C(Cc1ccccc1)NC(=O)C(CC(N)=O)NC(=O)c1ccc2ccccc2n1. References: Kupferschmidt H...
| Keywords: | Ro 31-8959 |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 127779-20-8 |
| MW: | 670.84 D |
From 34.00€
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Nelfinavir
Item number: TGM-T7779-100mg
Description: Nelfinavir (AG1341) is an antiretroviral drug used in the treatment of the human immunodeficiency virus (HIV) (Ki=2 nM). Nelfinavir is a broad-spectrum, anticancer agent. Target: HIV Protease. Smiles: Cc1c(O)cccc1C(=O)N[C@@H](CSc1ccccc1)[C@H](O)CN1C[C@H]2CCCC[C@H]2C[C@H]1C(=O)NC(C)(C)C. References:...
| Keywords: | AG1341 |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 159989-64-7 |
| MW: | 567.78 D |
From 37.00€
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