68 products were found matching "K15528"!
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Fatty Acid Amide Hydrolase (human, recombinant)
Item number: Cay10010183-100
Fatty acid amide hydrolase (FAAH) is a serine hydrolase with a major role in the hydrolysis of endocannabinoids. It is composed of an N-terminal transmembrane domain, a catalytic domain containing an amidase signature sequence, a polyproline sequence, and a monotopic membrane binding domain. FAAH is localized to...
| Keywords: | FAAH, FAAH1, Oleamide hydrolase 1, Oleamide hydrolase 1, Anandamide amidohydrolase 1, Anandamide amidohydrolase 1,... |
| Application: | Enzyme activity |
| MW: | 67,5 kD |
732.00€
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URB597
Item number: Cay10046-10
URB597 is a potent and selective inhibitor of fatty acid amide hydrolase (FAAH), the enzyme that hydrolyzes anandamide (AEA, Cay-90050) and other simple esters and amides with long unsaturated acyl chains (IC50 = 4.6 nM and 0.5 nM in brain membranes and intact neurons, respectively). URB597 exhibits both...
| Keywords: | (3'-(aminocarbonyl)[1,1'-biphenyl]-3-yl)-cyclohexylcarbamate |
| Application: | FAAH inhibitor |
| CAS | 546141-08-6 |
| MW: | 338.4 D |
From 44.00€
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PHOP
Item number: Cay71655-100
Fatty acid amide hydrolase (FAAH) is the enzyme responsible for hydrolysis and inactivation of fatty acid amides including anandamide and oleamide. PHOP is a potent FAAH inhibitor, exhibiting Ki values of 0.094 nM and 0.2 nM for the human and rat enzymes, respectively. Using a proteomics approach, PHOP was screened...
| Keywords: | CAY10402, Phenyl hexanoyl oxazolopyridine, 1-oxazolo[4,5-b]pyridin-2-yl-6-phenyl-1-hexanone |
| Application: | FAAH inhibitor |
| CAS | 288862-83-9 |
| MW: | 294.4 D |
From 67.00€
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Anti-Fatty Acid Amide Hydrolase
Item number: Cay101600-1
Fatty acid amide hydrolase (FAAH) is a serine hydrolase with a major role in the hydrolysis of endocannabinoids. It is composed of an N-terminal transmembrane domain, a catalytic domain containing an amidase signature sequence, a polyproline sequence, and a monotopic membrane binding domain. FAAH is localized to...
| Keywords: | Anti-Faah, Anti-Faah1, Anti-Anandamide amidase, Anti-Anandamide amidase, Anti-Oleamide hydrolase 1, Anti-Oleamide... |
| Application: | IHC, WB |
| Host: | Rabbit |
| Species reactivity: | human, rat, mouse, ferret |
431.00€
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4-Nonylphenylboronic acid
Item number: TGM-T7688-100mg
Description: 4-Nonylphenylboronic acid is a inhibitor of FAAH. Target: FAAH. Smiles: CCCCCCCCCc1ccc(cc1)B(O)O. References: Minkkila? A , Saario S M , Ka?Sna?Nen H , et al. Discovery of Boronic Acids as Novel and Potent Inhibitors of Fatty Acid Amide Hydrolase[J]. Journal of Medicinal Chemistry, 2008, 51(22):7057-7060.
| Application: | FAAH inhibitor |
| CAS | 256383-45-6 |
| MW: | 248.17 D |
From 30.00€
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URB937
Item number: TGM-T8646-100mg
Description: URB937 is an inhibitor of FAAH and increases anandamide levels(IC50 : 26.8 nM). Target: FAAH. Smiles: NC(=O)c1cccc(c1)-c1cc(OC(=O)NC2CCCCC2)ccc1O. References: Clapper J R , Moreno-Sanz G , Russo R , et al. Anandamide suppresses pain initiation through a peripheral endocannabinoid mechanism.[J]. Nature...
| Application: | FAAH inhibitor |
| CAS | 1357160-72-5 |
| MW: | 354.4 D |
From 42.00€
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(±)17(18)-EpETE-Ethanolamide
Item number: TGM-T85120-10mg
Description: (±)17(18)-EpETE-Ethanolamide, an omega-3 endocannabinoid epoxide, originates from eicosapentaenoic ethanolamide (EPEA) through cytochrome P450 (CYP) epoxygenases action and is decomposed by soluble epoxide hydrolase (sEH) and fatty acid amide hydrolase (FA, AH). Its endogenous synthesis occurs in...
| Keywords: | 17,18-epoxy-Eicosatetraenoic Acid Ethanolamide, (±)17(18)-EpETE-EA, 17,18-EEQ-EA, (±)17,18-EEQ-Ethanolamide |
| Application: | omega-3 endocannabinoid epoxide, soluble epoxide hydrolase (sEH) & FAAH substrate |
| CAS | 2123491-23-4 |
| MW: | 361.52 D |
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FAAH inhibitor 2
Item number: TGM-T84404-10mg
Description: FAAH Inhibitor 2 (Compound 17b) is an irreversible inhibitor of fatty acid amide hydrolase (FAAH), demonstrating an IC50 value of 0.153 µM [1]. Target: Others. Smiles: C(OC(NCCCCCCC/C=C\CCCCCCCC)=O)C=1C=CC=NC1
| Application: | FAAH inhibitor |
| CAS | 1450603-63-0 |
| MW: | 388.59 D |
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3-Decyl-5,5'-diphenyl-2-thioxo-4-imidazolidinone
Item number: TGM-T84521-10mg
Description: 3-Decyl-5,5'-diphenyl-2-thioxo-4-imidazolidinone (compound 45), having a pI50 of 5.89, shows promise as an inhibitor of fatty acid amide hydrolase (FAAH). Despite its activity, it demonstrates a lack of affinity for cannabinoid receptors CB(1) and CB(2) [1]. Target: Others. Smiles:...
| Application: | FAAH inhibitor |
| CAS | 875014-22-5 |
| MW: | 408.6 D |
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O-Arachidonoyl glycidol
Item number: TGM-T84523-10mg
Description: O-Arachidonoyl glycidol (compound 1), a 2-arachidonoylglycerol (2-AG) analog, effectively inhibits the hydrolysis of cytosolic 2-oleoylglycerol (2-OG) with an IC50 value of 4.5 µM, and also blocks 2-OG and anandamide hydrolysis in membrane fractions with IC50 values of 19 µM and 12 µM, respectively [1]....
| Application: | Fatty acid amide hydrolase inhibitor |
| CAS | 439146-24-4 |
| MW: | 360.53 D |
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CAY10435
Item number: TGM-T84554-10mg
Description: CAY10435, a beta-ketooxazapyridine and selective FAAH inhibitor, exhibits antimicrobial properties. It binds non-competitively to the FAAH of Dictyostelium discoideum, demonstrating a Kd value of 0.57 nM [1] [2]. Target: Others. Smiles: C(CCCCCCCCCCC)(=O)C1=NC=2C(O1)=CC=CN2
| Application: | FAAH inhibitor |
| CAS | 288862-73-7 |
| MW: | 302.41 D |
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URB-597
Item number: TGM-T6714-100mg
Description: URB-597 (FAAH Inhibitor II) is an effective, orally bioavailable FAAH inhibitor (IC50: 4.6 nM), and no effect on other cannabinoid-related targets. Target: FAAH, Autophagy, Mitophagy. Smiles: NC(=O)c1cccc(c1)-c1cccc(OC(=O)NC2CCCCC2)c1. References: Mor M, et al. J Med Chem, 2004, 47(21), 41998-52008.
| Keywords: | FAAH Inhibitor II, KDS-4103 |
| Application: | FAAH inhibitor |
| CAS | 546141-08-6 |
| MW: | 338.4 D |
From 34.00€
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