174 products were found matching "K05175"!
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Etomidate (CRM)
Item number: Cay41826-1
Etomidate (CRM) (Cay-41826) is a certified reference material categorized as an anesthetic. Etomidate has been associated with overdose and death. Formulations containing etomidate have been used as anesthetics.This product is intended for research and forensic applications.Formal Name:...
| Keywords: | (+)-Etomidate, (R)-Etomidate, d-Etomidate, R 16659, 1-[(1R)-1-phenylethyl]-1H-imidazole-5-carboxylic acid ethyl ester |
| Application: | Certified reference material, anesthetic |
| CAS | 33125-97-2 |
| MW: | 244.3 D |
180.00€
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Clomethiazole
Item number: TGM-T14983-100mg
Description: Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It also has the potential for treating convulsive status epilepticus. Chlormethiazole inhibits cytochrome P450 isoforms: CYP2A6 and CYP2E1 in human liver microsomes. Target: GABA Receptor, P450. Smiles:...
| Keywords: | 5-(2-CHLOROETHYL)-4-METHYLTHIAZOLE, Chlormethiazole, Distraneurin |
| Application: | Targets gamma-aminobutyric acid receptor subunit alpha (GABRA) |
| CAS | 533-45-9 |
| MW: | 161.65 D |
From 41.00€
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NS11394
Item number: TGM-T2067-1mg
Description: NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator, possesses a functional efficacy selectivity profile of alpha(5) > alpha(3) > alpha(2) > alpha(1) at GABA(A) alpha subunit-containing receptors. Target: GABA Receptor. Smiles: CC(C)(O)c1ccc2n(cnc2c1)-c1cccc(c1)-c1ccccc1C#N....
| Keywords: | NS 11394 |
| Application: | GABA(A) receptor positive allosteric modulator |
| CAS | 951650-22-9 |
| MW: | 353.42 D |
From 33.00€
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Thiomuscimol hydrobromide
Item number: TGM-T28965-10mg
Description: Thiomuscimol hydrobromide is an agonist of GABAA receptor. Target: Others. Smiles: C(N)C1=CC(=O)NS1
| Application: | GABA(A) receptor agonist |
| CAS | 62020-54-6 |
| MW: | 130.17 D |
From 151.00€
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Chlormethiazole edisylate
Item number: TGM-T27007-25mg
Description: Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic. Target: Others. Smiles: O=S(=O)(O)CCS(=O)(=O)O.ClCCC=1SC=NC1C. References: Harenko A. A comparison between chlormethiazole and nitrazepam as hypnotics in...
| Keywords: | Clomethiazole ethanedisulfonate, Heminevrin, Clomethiazole edisylate, Hemithiamine, Distraneurin |
| Application: | Targets gamma-aminobutyric acid receptor subunit alpha (GABRA) |
| CAS | 1867-58-9 |
| MW: | 351.85 D |
From 1,491.00€
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AZD7325
Item number: TGM-T7699-100mg
Description: AZD7325 (AZD-7325) is a GABA-Aalpha2,3 -selective receptor modulator. Target: GABA Receptor, P450. Smiles: CCCNC(=O)c1nnc2c(cccc2c1N)-c1c(F)cccc1OC. References: ProfileToshihiro Nomura, et al. Potentiating alpha2 subunit containing perisomatic GABAA receptors protects against seizures in a mouse model...
| Keywords: | AZD-7325 |
| Application: | Alpha2- / alpha3 subunit-containing GABAA receptor positive allosteric modulator |
| CAS | 942437-37-8 |
| MW: | 354.38 D |
From 63.00€
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Avermectin B1a
Item number: TGM-T7605-100mg
Description: Avermectin B1a is a macrocyclic lactone disaccharide anthelmintic agent . Target: Parasite, Antibiotic. Smiles:...
| Keywords: | Avamectin B1a, Abamectin B1a |
| Application: | Anthelmintic agent |
| CAS | 65195-55-3 |
| MW: | 873.08 D |
From 30.00€
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6-(4-Methoxyphenyl)-3-pyridazinamine
Item number: TGM-T7793-100mg
Description: 6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist. Target: GABA Receptor. Smiles: COC1=CC=C(C=C1)C1=CC=C(N)N=N1. References: Wermuth C G , Bourguignon J J , Schlewer G , et al. ChemInform Abstract: Synthesis and Structure-Activity Relationships of a Series of Aminopyridazine...
| Application: | GABAA receptor antagonist |
| CAS | 4776-87-8 |
| MW: | 201.22 D |
From 43.00€
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GABRA1 Protein, Human, Recombinant (His)
Item number: TGM-TMPH-01366-100ug
Description: GABRA1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 29.9 kDa and the accession number is P14867.
| Keywords: | GABRA1, GABA(A) receptor subunit alpha-1, Gamma-aminobutyric acid receptor subunit alpha-1 |
| MW: | 29.9 kD |
From 352.00€
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L-655708
Item number: TGM-TQ0151-10mg
Description: L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM. Target: GABA Receptor. Smiles: [H][C@@]12CCCN1C(=O)c1cc(OC)ccc1-n1cnc(C(=O)OCC)c21. References: Saab BJ, et al. Short-term memory impairment after isoflurane in mice is prevented by the alpha5...
| Application: | Nootropic GABA(A) receptor subunit alpha-5 ligand |
| CAS | 130477-52-0 |
| MW: | 341.36 D |
From 76.00€
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Lorediplon
Item number: TGM-TQ0023-100mg
Description: Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the alpha1-subunit, associated with promoting sleep. Target: GABA Receptor. Smiles: CN(C(C)=O)c1cc(ccc1F)-c1ccnc2c(cnn12)C(=O)c1cccs1. References: Horoszok L, et al. A single-dose, randomized,...
| Application: | GABRA1 ligand |
| CAS | 917393-39-6 |
| MW: | 394.42 D |
From 39.00€
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ONO-8590580
Item number: TGM-TQ0040-100mg
Description: ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA alpha5. Target: GABA Receptor. Smiles: Cc1c(F)c(Nc2ccc(cn2)-c2cn(C)cn2)cc2n(CC3CC3)cnc12. References: Kawaharada S, et al. ONO-8590580, a Novel GABAAalpha5 Negative Allosteric Modulator Enhances Long-Term Potentiation and Improves...
| Keywords: | CS-2894 |
| Application: | Alpha5 subunit-containing GABAA receptor (benzodiazepine binding site) negative allosteric modulator |
| CAS | 1802661-73-9 |
| MW: | 376.43 D |
From 59.00€
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