85 products were found matching "K04615"!
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CGP 55845 hydrochloride
Item number: TGM-T21759-10mg
Description: CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC50 of 6 nM, suitable for use in neurological research [1] [2]. Target: Others. Smiles: Cl.C[C@H](NC[C@H](O)CP(O)(=O)Cc1ccccc1)c1ccc(Cl)c(Cl)c1
| Application: | GABAB receptor antagonist |
| CAS | 149184-22-5 |
| MW: | 438.71 D |
From 671.00€
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CGP 35348
Item number: TGM-T21793-1mg
Description: CGP 35348 is a selective antagonist of GABAB receptor (EC50 = 34 µM). CGP 35348 can be used in studies of neuromuscular coordination and spatial learning after neonatal brain damage in albino mice. Target: GABA Receptor. Smiles: C(P(CCCN)(=O)O)(OCC)OCC. References: Q Gillani, et al. CGP 35348, GABA B...
| Application: | GABA(B) receptor antagonist |
| CAS | 123690-79-9 |
| MW: | 225.22 D |
From 45.00€
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Arbaclofen placarbil
Item number: TGM-T30118-100mg
Description: Arbaclofen placarbil( XP19986) is a GABA(B) receptor agonist.Arbaclofen Placarbil is a novel R-baclofen prodrug with improved absorption, distribution, metabolism, and elimination properties compared to R-baclofen. And it can reduce postprandial reflux in patients with gastroesophageal reflux disease....
| Keywords: | XP-19986, XP 19986, XP19986 |
| Application: | Targets gamma-aminobutyric acid type B receptor (GABBR) |
| CAS | 847353-30-4 |
| MW: | 399.87 D |
From 1,671.00€
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Valiloxibic acid
Item number: TGM-T39962-1mL
Description: Valiloxibic acid is a prodrug of gamma-Hydroxybutyric acid (GHB).GHB is a naturally occurring neurotransmitter and a psychoactive drug, it acts on the GHB receptor and is a weak agonist at the GABAB receptor. Target: Others. Smiles: CC(C)[C@H](N)C(=O)OCCCC(O)=O. References: Xiang, Jia-Ning, Xu, Xuesong,...
| Keywords: | XWL-008, Acidum valiloxibicum |
| Application: | Targets gamma-aminobutyric acid type B receptor (GABBR) |
| CAS | 238401-16-6 |
| MW: | 203.238 D |
From 52.00€
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rac-BHFF
Item number: TGM-T4176-100mg
Description: rac-BHFF ((R,S)-BHFF) is potent and selective GABA B receptor positive allosteric modulator that increases the potency and efficacy of GABA ( > 15-fold and > 149% respectively). It exhibits anxiolytic activity in vivo and is orally active. Target: GABA Receptor. Smiles:...
| Keywords: | (R,S)-BHFF |
| Application: | GABA(B) receptor positive allosteric modulator |
| CAS | 123557-91-5 |
| MW: | 330.34 D |
From 55.00€
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CGP52432
Item number: TGM-T4363-10mg
Description: CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM). Target: GABA Receptor. Smiles: C(NCCCP(C(OCC)OCC)(=O)O)C1=CC(Cl)=C(Cl)C=C1. References: Bonanno G,etal.GABA(B) receptors as potential targets for drugs able to prevent excessive excitatory amino acid transmission in the spinal...
| Keywords: | CGP 52432 |
| Application: | GABA(B) receptor antagonist |
| CAS | 139667-74-6 |
| MW: | 384.24 D |
From 34.00€
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Saclofen
Item number: TGM-T4440-100mg
Description: Saclofen is a sulfonic analog of the inhibitory neurotransmitter gamma-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 µM).1 This compound can be used to determine the functional roles for the GABAB receptor as a mediator of slow inhibitory postsynaptic...
| Application: | Competitive GABAB receptor antagonist |
| CAS | 125464-42-8 |
| MW: | 249.71 D |
From 52.00€
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CGP36216 hydrochloride
Item number: TGM-T84878-10mg
Description: CGP36216 hydrochloride acts as a selective antagonist at the presynaptic GABA receptor, specifically binding to the GABAB receptor with a Ki value of 0.3 µM. This compound is leveraged in research focused on anxiety and trauma-related disorders [1] [2]. Target: Others. Smiles: P(CCCN)(CC)(=O)O.Cl
| Application: | GABAB receptor antagonist |
| CAS | 1781834-71-6 |
| MW: | 187.6 D |
Please request pricing for this article.
Baclofen-d4
Item number: TGM-TMIJ-0314-1mg
Description: Baclofen-d4 is a deuterated compound of Baclofen. Baclofen has a CAS number of 1134-47-0. Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing Baclofen acts as a gamma-aminobutyric acid (GABA) agonist...
| Application: | GC-MS, LC-MS, internal standard, GABA-B receptor agonist |
| CAS | 1189938-30-4 |
| MW: | 217.69 D |
Please request pricing for this article.
(R)-baclofen
Item number: TGM-T6355-100mg
Description: (R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity. Target: GABA Receptor. Smiles: NC[C@H](CC(O)=O)c1ccc(Cl)cc1. References: Falch E, et al. J Neurochem, 1986, 47(3), 898-903.
| Keywords: | Arbaclofen, STX209 |
| Application: | Targets gamma-aminobutyric acid type B receptor (GABBR) |
| CAS | 69308-37-8 |
| MW: | 213.66 D |
From 34.00€
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(R)-Baclofen hydrochloride
Item number: TGM-T17306-10mg
Description: Arbaclofen hydrochloride, a Gamma-Aminobutyric Acid derivative, is a specific agonist of GABA-B receptors, it is used to treat spasticity, especially that due to spinal cord damage. It acts at spinal and supraspinal sites, generally reduces excitatory transmission. Target: GABA Receptor. Smiles:...
| Keywords: | Arbaclofen hydrochloride |
| Application: | GABA(B) receptor agonist |
| CAS | 63701-55-3 |
| MW: | 250.12 D |
From 88.00€
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CGP 36742
Item number: TGM-T14938-2mg
Description: CGP 36742 is a selective antagonist of the GABAB receptor that can penetrate the blood-brain barrier after peripheral administration (IC50: 32 µM). It is useful in the treatment of depression. Target: GABA Receptor. Smiles: P(CCCC)(CCCN)(=O)O. References: Nowak G, et al. Antidepressant-like activity of...
| Keywords: | SGS-742 |
| Application: | GABAB receptor antagonist |
| CAS | 123690-78-8 |
| MW: | 179.2 D |
83.00€
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