84 products were found matching "K04280"!
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Gonadotropin-releasing hormone II receptor (GNRHR2),...
Item number: CSB-CF856800MOW.100
Organism: Macaca mulatta (Rhesus macaque). Source: in vitro E.coli expression system. Expression Region: 1-379aa. Protein Length: Full Length. Tag Info: N-terminal 6xHis-tagged. Target Protein Sequence: MSAGNGTPWG SAAGEESWAA SGVAVEGSEL PTFSAAAKVR VGVTIVLFVS SAGGNLAVLW SVTRPQPSQL RPSPVRTLFA HLAAADLLVT FVVMPLDATW...
| Keywords: | GNRHR2, GnRH-II-R, GnRH II receptor, Type II GnRH receptor, Gonadotropin-releasing hormone II receptor |
| Application: | Activity not tested |
| Expressed in: | E.coli in vitro |
| Origin: | Rhesus macaque |
| MW: | 42.4 kD |
From 1,458.00€
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LHRH Acetate Salt
Item number: LKT-L302690.100
Luteinizing hormone-releasing hormone (LHRH or Gonadotropin-releasing hormone [GnRH]) is an endogenous peptide hormone that binds the GnRH receptor, stimulating secretion of reproductive hormones (such as luteinizing hormone [LH ] and follicle-stimulating hormone [FSH]) from the pituitary gland. Analogs of GnRH are...
| Keywords: | Gonadorelin, Gonadorelin acetate salt, Luliberin, GnRH, LH-RH, human, pEHWSYGLRPG-NH3 |
| Application: | Endogenous peptide hormone, involved in secretion of reproductive hormones, GnRH agonist. |
| CAS | 33515-09-2 |
| MW: | 1182.31 D |
From 360.00€
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Nafarelin acetate(76932-56-4 free base)
Item number: TGM-T21309-5mg
Description: Nafarelin acetate(76932-56-4 free base) (RS-94991-298) is a GnRH agonist that acts as an analog of GnRH. Nafarelin acetate(76932-56-4 free base) causes a decrease in the pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH). It may be used in the treatment...
| Keywords: | RS-94991-298, Synarel, Nafarelin acetate, Nafarelin acetate hydrate |
| Application: | Gonadotropin-releasing hormone receptor agonist |
| CAS | 76932-60-0 |
| MW: | 1400.56 D |
From 49.00€
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Relugolix
Item number: TGM-T3630-100mg
Description: Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential antineoplastic activity. Relugolix competitively binds to and blocks the GnRH receptor in the anterior pituitary gland, which both...
| Keywords: | RVT-601, TAK-385 |
| Application: | Targets gonadotropin-releasing hormone receptor (GNRHR) |
| CAS | 737789-87-6 |
| MW: | 623.63 D |
From 31.00€
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Linzagolix
Item number: TGM-T27837-10mg
Description: Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei Pharmaceutical and ObsEva for the treatment of uterine fibroids, endometriosis, and adenomyosis. As of December 2020, it is under review for...
| Application: | Targets gonadotropin-releasing hormone receptor (GNRHR) |
| CAS | 935283-04-8 |
| MW: | 508.42 D |
From 37.00€
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Sufugolix
Item number: TGM-T3538-100mg
Description: Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone (LHRH) receptor antagonist. Target: LHRH. Smiles: CONC(=O)Nc1ccc(cc1)-c1sc2n(Cc3c(F)cccc3F)c(=O)n(-c3ccccc3)c(=O)c2c1CN(C)Cc1ccccc1. References: Sasaki S, et al. Discovery of a thieno[2,3-d]pyrimidine-2,4-dione...
| Keywords: | TAK-013 |
| Application: | Gonadotropin-releasing hormone receptor (GnRHR) antagonist |
| CAS | 308831-61-0 |
| MW: | 667.72 D |
From 37.00€
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Goserelin acetate
Item number: TGM-T4102-100mg
Description: Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer. Target: Apoptosis, GNRH Receptor. Smiles:...
| Keywords: | Zoladex, Fertilan, ICI-118630 acetate |
| Application: | Targets gonadotropin-releasing hormone receptor (GNRHR) |
| CAS | 145781-92-6 |
| MW: | 1329.46 D |
From 42.00€
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Gonadorelin HCl
Item number: TGM-T5015L2-100mg
Description: Gonadorelin HCl, as a decapeptide, can stimulate the synthesis and secretion of both pituitary gonadotropins, LUTEINIZING HORMONE, and FOLLICLE STIMULATING HORMONE. Target: Others. Smiles:...
| Keywords: | Factrel, AY-24,031, AY24,031, AY 24,031, LH-RH hydrochloride, Gonadorelin hydrochloride |
| Application: | Targets gonadotropin-releasing hormone receptor (GNRHR) |
| CAS | 51952-41-1 |
| MW: | 1218.77 D |
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Elagolix sodium
Item number: TGM-T5031-100mg
Description: Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively). Target: GNRH Receptor. Smiles: [Na+].COc1cccc(c1F)-c1c(C)n(Cc2c(F)cccc2C(F)(F)F)c(=O)n(C[C@H](NCCCC([O-])=O)c2ccccc2)c1=O. References: Barra F, Scala C, Ferrero S2.Elagolix sodium...
| Keywords: | NBI-56418 sodium |
| Application: | Targets gonadotropin-releasing hormone receptor (GNRHR) |
| CAS | 832720-36-2 |
| MW: | 653.57 D |
From 40.00€
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Cetrorelix Acetate
Item number: TGM-T5520-100mg
Description: Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM. Target: GNRH Receptor. Smiles:...
| Keywords: | Cetrorelix |
| Application: | Targets gonadotropin-releasing hormone receptor (GNRHR) |
| CAS | 145672-81-7 |
| MW: | 1491.11 D |
From 42.00€
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Cetrorelix diacetate
Item number: TGM-T5520L-100mg
Description: Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the production and action of luteinizing hormone (LH) and follicle-stimulating hormone (FSH). Target: GNRH Receptor. Smiles:...
| Keywords: | SB-075 acetate, NS-75A, Cetrorelix acetate, SB-075 diacetate, NS-75A diacetate |
| Application: | GnRH inhibitor |
| CAS | 130143-01-0 |
| MW: | 1551.17 D |
From 48.00€
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Nafarelin acetate hydrate
Item number: TGM-T68525-100mg
Description: Nafarelin is a gonadotropin-releasing hormone agonist (GnRH agonist) which acts as an analog of GnRH. Nafarelin increases the release of FSH and LH by the anterior pituitary, which in turn leads to an increase of estrogen/progesterone. When administered, Nafarelin has the purpose of causing increase...
| Application: | Targets gonadotropin-releasing hormone receptor (GNRHR) |
| CAS | 86220-42-0 |
| MW: | 1400.563 D |
From 2,873.00€
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