44 products were found matching "K04228"!
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Argipressin
Item number: TGM-T7434-10mg
Description: Argipressin (Vasopressin) is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth muscle cells and neonatal rat cardiomyocytes, respectively. Target: Vasopressin...
| Keywords: | Vasopressin, Arg8-vasopressin, AVP |
| Application: | Targets arginine vasopressin receptor 2 (AVPR2) |
| CAS | 113-79-1 |
| MW: | 1084.23 D |
From 46.00€
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LIXIVAPTAN
Item number: TGM-T7303-100mg
Description: Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM). Target: Vasopressin Receptor. Smiles: Cc1ccc(F)cc1C(=O)Nc1ccc(C(=O)N2Cc3cccn3Cc3ccccc23)c(Cl)c1. References: Wang X, Constans MM, Chebib FT.et al.Effect of a Vasopressin V2 Receptor Antagonist on...
| Keywords: | WAY-VPA 985, VPA-985 |
| Application: | Targets arginine vasopressin receptor 2 (AVPR2) |
| CAS | 168079-32-1 |
| MW: | 473.93 D |
From 37.00€
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AVPR2 Protein, Pig, Recombinant (His & SUMO)
Item number: TGM-TMPH-03132-100ug
Description: Receptor for arginine vasopressin. The activity of this receptor is mediated by G proteins which activate adenylate cyclase. Involved in renal water reabsorption. AVPR2 Protein, Pig, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight...
| Keywords: | AVPR V2, Renal-type arginine vasopressin receptor, Antidiuretic hormone receptor, V2R, AVPR2, Vasopressin V2 receptor |
| MW: | 24.7 kD |
From 359.00€
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Ornipressin
Item number: TGM-TP1049-10mg
Description: Ornipressin is a vasoconstrictor, haemostatic and renal agent. Smiles: NCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CSSC[C@H](N)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N1)C(=O)NCC(N)=O. References: Fruhstorfer H, et al. Dose-response relation of...
| Keywords: | POR-8 |
| Application: | Targets arginine vasopressin receptor 2 (AVPR2) |
| CAS | 3397-23-7 |
| MW: | 1042.19 D |
From 58.00€
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Lysipressin
Item number: TGM-T11918-10mg
Description: Lysipressin ([Lys8]-Vasopressin), Induces contraction of the rabbit urinary bladder smooth muscle, activate adenylate-cyclase. Lysipressin is Antidiuretic hormone that have been found in pigs and some marsupial families. Target: Others. Smiles:...
| Keywords: | Lysine vasopressin, [Lys8]-Vasopressin |
| Application: | Targets arginine vasopressin receptor 2 (AVPR2) |
| CAS | 50-57-7 |
| MW: | 1056.22 D |
From 100.00€
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Terlipressin
Item number: TGM-T13920-500mg
Description: Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells. Target: Others. Smiles:...
| Application: | Targets arginine vasopressin receptor 2 (AVPR2) |
| CAS | 14636-12-5 |
| MW: | 1227.37 D |
1,214.00€
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Anti-AVPR2
Item number: CSB-PA222915.100
Host Species: Rabbit. Isotype: IgG. Buffer: Liquid in PBS containing 50% glycerol, 0.5% BSA and 0.02% sodium azide. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: The antibody was affinity-purified from rabbit antiserum by affinity-chromatography using epitope-specific...
| Keywords: | Anti-V2R, Anti-ADHR, Anti-AVPR2, Anti-AVPR V2, Anti-Vasopressin V2 receptor, Anti-Antidiuretic hormone receptor,... |
| Application: | ELISA, WB |
| Host: | Rabbit |
| Species reactivity: | human, mouse |
From 126.00€
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Anti-AVPR2
Item number: CSB-PA987235.100
Host Species: Rabbit. Isotype: IgG. Buffer: -20°C, pH7.4 PBS, 0.05% NaN3, 40% Glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Antigen affinity purification. Target Name: AVPR2. Antigen Species: Human
| Keywords: | Anti-V2R, Anti-ADHR, Anti-AVPR2, Anti-AVPR V2, Anti-Vasopressin V2 receptor, Anti-Antidiuretic hormone receptor,... |
| Application: | ELISA, IHC |
| Host: | Rabbit |
| Species reactivity: | human |
From 167.00€
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Vasopressin V2 receptor (AVPR2), partial, swine, recombinant
Item number: CSB-EP002470PI.1
Organism: Sus scrofa (Pig). Source: E.coli. Expression Region: 292-370aa. Protein Length: Partial. Tag Info: N-terminal 6xHis-SUMO-tagged. Target Protein Sequence: WSVWDPKAPR EGPPFVLLML LASLNSCTNP WIYASFSSSI SSELRSLLCC PRRRTPPSLR PQEESCATAS SFSARDTSS. Purity: Greater than 90% as determined by SDS-PAGE. Endotoxin:...
| Keywords: | V2R, AVPR2, AVPR V2, Vasopressin V2 receptor, Antidiuretic hormone receptor, Renal-type arginine vasopressin receptor,... |
| Application: | Activity not tested |
| Expressed in: | E.coli |
| Origin: | swine |
| MW: | 24.7 kD |
From 364.00€
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Tolvaptan
Item number: LKT-T5847.500
A potent human vasopressin V2-receptor antagonist. It increases serum sodium concentration in patients with euvolemic or hypervolemic hyponatremia.
| Keywords: | OPC-41061, N-(4-(((5R)-7-chloro-5-hydroxy-2,3,4,5-tetrahydro-1H-1-benzazepin-1-yl)carbonyl)-3-methylphenyl)-2-methylbenzamide |
| Application: | Vasopressin V2-receptor antagonist |
| CAS | 150683-30-0 |
| MW: | 448,94 D |
From 149.00€
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Tolvaptan
Item number: Cay19691-1
Tolvaptan is a nonpeptide vasopressin V2 receptor antagonist (IC50 = 3 nM for rat receptor) and a diuretic agent. It is selective for V2 over V1 receptors (IC50 = 0.58 µM). Tolvaptan increases urine volume by 3-fold in rats when administered at a dose of 0.54 mg/kg. It also reduces left ventricular end-systolic...
| Keywords: | OPC 41061, N-[4-[(7-chloro-2,3,4,5-tetrahydro-5-hydroxy-1H-1-benzazepin-1-yl)carbonyl]-3-methylphenyl]-2-methyl-benzamide |
| Application: | AVPR2 antagonist |
| CAS | 150683-30-0 |
| MW: | 448.9 D |
From 44.00€
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Conivaptan (hydrochloride)
Item number: Cay23728-5
Conivaptan is an antagonist of the arginine vasopressin (AVP) receptors V1A and V2 (Kis = 0.48 and 3.04 nM for rat liver V1A and kidney V2, respectively). It also competitively inhibits oxytocin binding to rat uterine oxytocin receptors (Ki = 44 nM) but has no effect on AVP binding to anterior pituitary V1B...
| Keywords: | YM-087, N-[4-[(4,5-dihydro-2-methylimidazo[4,5-d][1]benzazepin-6(1H)-yl)carbonyl]phenyl]-[1,1'-biphenyl]-2-carboxamide,... |
| Application: | Vasopressin receptor antagonist |
| CAS | 168626-94-6 |
| MW: | 535 D |
From 94.00€
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