329 products were found matching "K04215"!

(±)-Methadone-d3 (CRM) (Cay-35882) is intended for use as an internal standard for the quantification of methadone by GC- or LC-MS. (±)-Methadone is categorized as an opioid. It has analgesic activity. Formulations containing (±)-methadone have been used in the treatment of opioid addiction. (±)-Methadone-d3 is...

Organism: Homo sapiens (Human). Source: in vitro E.coli expression system. Expression Region: 1-400aa. Protein Length: Full Length. Tag Info: N-terminal 10xHis-tagged. Target Protein Sequence: MDSSAAPTNA SNCTDALAYS SCSPAPSPGS WVNLSHLDGN LSDPCGPNRT DLGGRDSLCP PTGSPSMITA ITIMALYSIV CVVGLFGNFL VMYVIVRYTK MKTATNIYIF...

(±)-Methadone-d9 (CRM) (Cay-39479) is intended for use as an internal standard for the quantification of methadone by GC- or LC-MS. (±)-Methadone is categorized as an opioid. It has analgesic activity. Formulations containing (±)-methadone have been used in the treatment of opioid addiction. (±)-Methadone-d9 is...

SR 17018 is an orally bioavailable and brain-penetrant agonist of µ-opioid receptors. It is functionally selective for G protein-coupled receptor signaling (EC50 = 97 nM for GTPgammaS binding in CHO cells expressing µ-opioid receptors) over beta-arrestin 2 recruitment (EC50 = >10,000 nM) at the µ-opioid receptor. SR...

In 1X PBS, pH 7.4, with 0.09% sodium azide. OPRM1 is the mu opioid receptor, which is the primary site of action for the most commonly used opioids, including morphine, heroin, fentanyl, and methadone. It is also the primary receptor for endogenous opioid peptides beta-endorphin and the enkephalins. The OPRM1...

Small compounds (drugs or peptides) are not sufficiently complex by themselves to induce an immune response or be processed in a manner that elicits production of specific antibodies. For antibody production to be successful with small antigens, they must be chemically conjugated with immunogenic carrier proteins...

alpha-methyl Butyryl fentanyl (hydrochloride) (Cay-20818) is an analytical reference standard that is structurally similar to known opioids. alpha-methyl Butyryl fentanyl is regulated as a Schedule I compound in the United States. This product is intended for research and forensic applications.Formal Name:...

Mitraciliatine is an alkaloid that has been found in M. speciosa (Kratom in Thai) and is a µ-opioid receptor (MOR) partial agonist and kappa-opioid receptor (KOR) agonist. It is selective for MOR and KOR over the delta-opioid receptor (DOR, EC50s = 228, 218, and >1,000 nM, respectively, for the mouse receptors in a...

The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human OPRM1. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Human OPRM1. Next,...

Meptazinol (hydrochloride) (Cay-39657) is an analytical reference standard categorized as an opioid. Meptazinol induces analgesia in mice. This product is intended for research and forensic applications.Formal Name: 3-(3-ethylhexahydro-1-methyl-1H-azepin-3-yl)-phenol, monohydrochloride. CAS Number: 59263-76-2....

N-didesmethyl Loperamide is an active metabolite of the peripheral µ1-opioid receptor agonist loperamide. It inhibits electricity-induced contractions in isolated guinea pig myenteric plexus (IC50 = 370 nM). N-didesmethyl Loperamide sensitizes a chloroquine-resistant P. falciparum strain to chloroquine (EC50 = 482...

A mu-opioid agonist that is an antidiarrhoeal drug which inhibits intestinal motility and secretion. It has been shown to suppress the calcium-influx in dorsal root ganglion neurons.