241 products were found matching "K04157"!
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Clozapine (hydrochloride)
Item number: Cay25779-25
Clozapine is a partial agonist of the serotonin (5-HT) receptor subtype 5-HT1A (Ki = 180 nM). It also binds to the 5-HT2A, 5-HT2C, 5-HT3, 5-HT6, and 5-HT7 receptors (Kis = 3.3, 13, 110, 4, and 21 nM, respectively), as well as the histamine H1 and alpha1-adrenergic receptors (Kis = 2.1 and 23 nM, respectively). It...
| Keywords: | 8-chloro-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine, dihydrochloride |
| Application: | Atypical antipsychotic, multi-acting receptor targeted antipsychotic (MARTA) |
| CAS | 2711603-38-0 |
| MW: | 399.7 D |
133.00€
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(+)-Fenfluramine (hydrochloride)
Item number: Cay39830-100
(+)-Fenfluramine is an agonist of the serotonin (5-HT) receptor subtypes 5-HT2B and 5-HT2C. It induces serotonin release from superfused midbrain synaptosome preparations isolated from wild-type mice, but not 5-HT2B-/- mice, when used at concentrations of 0.5 or 1 µM. (+)-Fenfluramine (3 or 10 mg/kg) reduces food...
| Keywords: | Dexfenfluramine, N-ethyl-alpha-methyl-3-(trifluoromethyl)-benzeneethanamine, monohydrochloride |
| Application: | 5-HT2B / 5-HT2C receptor agonist |
| CAS | 3239-45-0 |
| MW: | 267.7 D |
243.00€
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Risperidone (CRM)
Item number: Cay40163-1
Risperidone (CRM) (Cay-40163) is a certified reference material classified as an atypical antipsychotic. Risperidone has been abused recreationally. Formulations containing risperidone have been used in the treatment of schizophrenia and bipolar disorder. This product is intended for research and forensic...
| Keywords: | Apexidone, Psychodal, R 64766,... |
| Application: | Certified reference material, atypical antipsychotic, serotonin-dopamine antagonists (SDA) |
| CAS | 106266-06-2 |
| MW: | 410.5 D |
134.00€
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Paliperidone (CRM)
Item number: Cay40387-1
Paliperidone (CRM) (Cay-40387) is a certified reference material categorized as an atypical antipsychotic. Paliperidone is an active metabolite of risperidone. It has anticonvulsant, antinociceptive, and antidepressant-like activities in rats. Paliperidone also inhibits apomorphine-induced agitation and stereotypy...
| Keywords: | 9-hydroxy Risperidone, RO76477,... |
| Application: | Certified reference material, atypical antipsychotic |
| CAS | 144598-75-4 |
| MW: | 426.5 D |
252.00€
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5-hydroxytryptamine receptor 2C (Htr2c), recombinant...
Item number: CSB-CF010889MO.100
Organism: Mus musculus (Mouse). Source: in vitro E.coli expression system. Expression Region: 33-459aa. Protein Length: Full Length of Mature Protein. Tag Info: N-terminal 10xHis-tagged. Target Protein Sequence: IVTDTFNSSD GGRLFQFPDG VQNWPALSIV VIIIMTIGGN ILVIMAVSME KKLHNATNYF LMSLAIADML VGLLVMPLSL LAILYDYVWP...
| Keywords: | Htr2c, 5ht1c, 5-HT1C, 5-HT2C, 5-HT-2C, 5-HT-1C, 5-HTR2C, Serotonin receptor 2C, 5-hydroxytryptamine receptor 2C,... |
| Application: | Activity not tested |
| Expressed in: | E.coli in vitro |
| Origin: | mouse |
| MW: | 54.6 kD |
From 1,458.00€
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Clozapine N-oxide
Item number: LKT-C4759.25
Metabolite of clozapine. It is 5-HT2 serotonin receptor antagonist.
| Application: | 5-HT2 serotonin receptor antagonist |
| CAS | 34233-69-7 |
| MW: | 342,82 D |
From 274.00€
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lurasidone-d8
Item number: TGM-TMIH-0313-10mg
Description: lurasidone-d8 is a deuterated compound of lurasidone. Smiles: [2H]C1([2H])N(C[C@@H]2CCCC[C@H]2CN2C(=O)[C@H]3[C@@H]4CC[C@@H](C4)[C@H]3C2=O)C([2H])([2H])C([2H])([2H])N(C2=NSC3=CC=CC=C23)C1([2H])[2H]
| Application: | GC-MS, LC-MS, internal standard |
| CAS | 1132654-54-6 |
| MW: | 500.73 D |
From 887.00€
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Paliperidone-d4
Item number: TGM-TMIH-0420-10mg
Description: Paliperidone-d4 is a deuterated compound of Paliperidone. Paliperidone has a CAS number of 144598-75-4. Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the primary active metabolite of the older...
| Application: | GC-MS, LC-MS, internal standard, quantification, Dopamine D2/3-receptor / 5-HT2A-receptor antagonist |
| CAS | 1020719-55-4 |
| MW: | 430.51 D |
From 592.00€
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Quetiapine-d8 Fumarate
Item number: TGM-TMIJ-0315-1mg
Description: Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression. Smiles:...
| Application: | GC-MS, LC-MS, internal standard, quantification, multiple receptor antagonist |
| CAS | 1185247-12-4 |
| MW: | 507.63 D |
Please request pricing for this article.
CP-809101
Item number: TGM-TQ0130-10mg
Description: CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors). Target: 5-HT Receptor. Smiles: O(CC1=CC(Cl)=CC=C1)C=2N=C(C=NC2)N3CCNCC3. References: Higgins GA, Silenieks LB, Lau W, et al. Evaluation of chemically diverse 5-HT2C receptor...
| Application: | Potent 5-HT2C receptor agonist |
| CAS | 479683-64-2 |
| MW: | 304.77 D |
From 233.00€
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Naftidrofuryl
Item number: TGM-T25848-100mg
Description: Naftidrofuryl is used in the management of peripheral and cerebral vascular disorders. It is claimed to enhance cellular oxidative capacity and to be spasmolytic. Target: Others. Smiles: C(C(CC1CCCO1)C(OCCN(CC)CC)=O)C=2C3=C(C=CC2)C=CC=C3. References: de Backer TL, Vander Stichele R, Lehert P, Van Bortel...
| Application: | Targets 5-hydroxytryptamine receptor 2 (HTR2) |
| CAS | 31329-57-4 |
| MW: | 383.52 D |
From 1,671.00€
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Metrenperone
Item number: TGM-T25806-100mg
Description: Metrenperone is used as a S(2)-receptor blocker. Target: Others. Smiles: O=C1N2C(=NC(C)=C1CCN3CCC(C(=O)C4=CC=C(F)C=C4)CC3)C=CC(C)=C2. References: Oryan A, Silver IA, Goodship AE. Metrenperone enhances collagen turnover and remodeling in the early stages of healing of tendon injury in rabbit. Arch Orthop...
| Keywords: | R 50970, R-50970, R50970 |
| Application: | Targets 5-hydroxytryptamine receptor 2 (HTR2) |
| CAS | 81043-56-3 |
| MW: | 407.48 D |
From 1,520.00€
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