- Search results for K04150
Cookie preferences
This website uses cookies, which are necessary for the technical operation of the website and are always set. Other cookies, which increase the comfort when using this website, are used for direct advertising or to facilitate interaction with other websites and social networks, are only set with your consent.
Configuration
Technically required
These cookies are necessary for the basic functions of the shop.
"Allow all cookies" cookie
"Decline all cookies" cookie
CSRF token
Cookie preferences
Currency change
Customer-specific caching
FACT-Finder tracking
Individual prices
Selected shop
Session
Comfort functions
These cookies are used to make the shopping experience even more appealing, for example for the recognition of the visitor.
Note
Show the facebook fanpage in the right blod sidebar
Statistics & Tracking
Affiliate program
Conversion and usertracking via Google Tag Manager
Track device being used
31 products were found matching "K04150"!
Close filters
Filter by:
No results were found for the filter!
Item number: Cay18743-5
Cimetidine is a histamine H2 receptor antagonist (Ki = 0.6 µM). It also acts as an inverse agonist, inhibiting basal cAMP production in CHO cells expressing recombinant H2 receptors (IC50 = 1.2 µM). Cimetidine inhibits histamine-induced acid secretion from isolated bullfrog gastric mucosa (IC50 = 16 µM). In vivo, it...
Keywords: | NSC 335308, SKF 92334, N-cyano-N''-methyl-N'-[2-[[(4-methyl-1H-imidazol-5-yl)methyl]thio]ethyl]-guanidine |
Application: | H2-receptor antagonist |
CAS | 51481-61-9 |
MW: | 252.3 D |
From 48.00€
*
Item number: Cay16939-1
Ranitidine is a histamine H2 receptor antagonist. It reverses histamine-induced relaxation of isolated rat uterine horn (pA2 = 6.9) as well as histamine-induced increases in contraction frequency in isolated guinea pig right atrium (pA2 = 7.2). Ranitidine (0.03-3 mg/kg, i.v.) inhibits histamine-and...
Keywords: | N'-[2-[[[5-[(dimethylamino)methyl]-2-furanyl]methyl]thio]ethyl]-N-methyl-2-nitro-1,1-ethenediamine, monohydrochloride |
Application: | H2-receptor antagonist |
CAS | 66357-59-3 |
MW: | 350.9 D |
From 43.00€
*
Item number: Cay33828-1
Histamine is a biogenic amine. It is produced from histidine in basophils, mast cells, gastric enterochromaffin-like (ECL) cells, and histaminergic neurons by histidine decarboxylase (HDC). Histamine activates the G protein-coupled histamine H1-4 receptors to regulate allergic and inflammatory responses, gastric...
Keywords: | NSC 33792, 1H-imidazole-5-ethanamine |
Application: | Biogenic amine, histamine H1-4 receptor agonist |
CAS | 51-45-6 |
MW: | 111.1 D |
From 97.00€
*
Item number: Cay21248-500
Roxatidine acetate is a competitive histamine H2 receptor antagonist that upon oral absorption is rapidly converted to its active metabolite roxatidine. By inhibiting the binding of histamine to H2 receptors, roxatidine reduces both intracellular cAMP concentrations and gastric acid secretion by parietal...
Keywords: | HOE 760, TZU-0460, 2-(acetyloxy)-N-[3-[3-(1-piperidinylmethyl)phenoxy]propyl]-acetamide, monohydrochloride |
Application: | H2 receptor antagonist |
CAS | 93793-83-0 |
MW: | 384.9 D |
From 43.00€
*
Item number: Cay23828-1
Famotidine is a histamine H2 receptor antagonist with a Ki value of 12 nM in fractionated guinea pig cerebral cortex membranes. It is selective for H2 over H1 and muscarinic receptors (Kis = 4 and 28 µM, respectively, in bovine cerebral cortex). Famotidine inhibits histamine-induced acid secretion in isolated canine...
Keywords: | MK-208, YM-11170, 3-[[[2-[(aminoiminomethyl)amino]-4-thiazolyl]methyl]thio]-N-(aminosulfonyl)-propanimidamide |
Application: | Histamine receptor H2 antagonist |
CAS | 76824-35-6 |
MW: | 337.5 D |
From 43.00€
*
Item number: Cay29418-50
Dimaprit is a histamine H2 receptor agonist with a Ki value of 44 µM in guinea pig right atrium. It is selective for histamine H2 over H1 and H3 receptors with relative potencies of 71, A. suum extract, which is not affected by pretreatment with mepyramine (Cay-20978), an H1 receptor inverse agonist, or cimetidine...
Keywords: | carbamimidothioic acid, 3-(dimethylamino)propyl ester, dihydrochloride |
Application: | Histamine H2 receptor agonist |
CAS | 23256-33-9 |
MW: | 234.2 D |
From 90.00€
*
Item number: Cay36111-1
Roxatidine is a histamine H2 receptor antagonist and major active metabolite of roxatidine acetate (Cay-21248). Roxatidine reduces histamine-induced adenylate cyclase production in guinea pig parietal cells (IC50 = 0.8 µM). It inhibits histamine-induced hydrogen ion accumulation in the same cells (pA2 = 7.03)....
Keywords: | 2-hydroxy-N-[3-[3-(1-piperidinylmethyl)phenoxy]propyl]-acetamide |
Application: | Histamine H2 receptor antagonist, Major active roxatidine acetate metabolite |
CAS | 78273-80-0 |
MW: | 306.4 D |
From 54.00€
*
Item number: ARG63821.100
Protein function: The H2 subclass of histamine receptors mediates gastric acid secretion. Also appears to regulate gastrointestinal motility and intestinal secretion. Possible role in regulating cell growth and differentiation. The activity of this receptor is mediated by G proteins which activate adenylyl cyclase...
Keywords: | Anti-H2R, Anti-HRH2, Anti-HH2R, Anti-Gastric receptor I, Anti-Histamine H2 receptor |
Application: | ELISA, IHC (paraffin) |
Host: | Goat |
Species reactivity: | human |
784.00€
*
Item number: LKT-N3496.10
A H2-receptor antagonist, found to be a potent inhibitor of gastric acid secretion.
Application: | H2-receptor antagonist |
CAS | 76963-41-2 |
MW: | 331,46 D |
From 94.00€
*
Item number: Cay18861-10
Histamine H2 receptors mediate gastric acid secretion by coupling to Galphas proteins and increasing cAMP formation. Nizatidine is a histamine H2 receptor antagonist that decreases gastric acid secretion (ED50 = 0.9 µM in isolated gastric mucosa of bullfrog and ED50s = 1.383 and 0.08 µmol/kg in rats and dogs,...
Keywords: | LY139037, N'-[2-[[[2-[(dimethylamino)methyl]-4-thiazolyl]methyl]thio]ethyl]-N-methyl-2-nitro-1,1-ethenediamine |
Application: | H2-receptor antagonist |
CAS | 76963-41-2 |
MW: | 331.5 D |
From 60.00€
*
Item number: LKT-R5894.1
A histamine H2-receptor antagonist used in ulcer treatment. It is found to inhibit platelet function in vitro.
Application: | H2-receptor antagonist |
CAS | 93793-83-0 |
MW: | 384,9 D |
From 149.00€
*
Item number: Cay29050-1
Cimetidine-d3 is intended for use as an internal standard for the quantification of cimetidine (Cay-18743) by GC- or LC-MS. Cimetidine is a histamine H2 receptor antagonist (Ki = 0.6 µM). It also acts as an inverse agonist, inhibiting basal cAMP production in CHO cells expressing recombinant H2 receptors (IC50 = 1.2...
Keywords: | N-cyano-N''-methyl-d3-N'-[2-[[(4-methyl-1H-imidazol-5-yl)methyl]thio]ethyl]-guanidine |
Application: | GC-MS, LC-MS, internal standard, quantification, H2-receptor antagonist |
CAS | 1185237-29-9 |
MW: | 255.4 D |
417.00€
*