173 products were found matching "K04149"!
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Norastemizole
Item number: Cay41828-1
Norastemizole is a histamine H1 receptor antagonist (IC50 = 4.1 nM) and an active metabolite of the histamine H1 receptor antagonist and ether-a-go-go (ERG) channel blocker astemizole (Cay-16967). It is formed from astemizole by the cytochrome P450 (CYP) isoform 3A4 (CYP3A4). Norastemizole also inhibits currents in...
| Keywords: | Tecastemizole, 1-[(4-fluorophenyl)methyl]-N-4-piperidinyl-1H-benzimidazol-2-amine |
| Application: | Astemizole active metabolite, histamine H1 receptor antagonist |
| CAS | 75970-99-9 |
| MW: | 324.4 D |
From 52.00€
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Promethazine-d3 (hydrochloride) (CRM)
Item number: Cay39606-100
Promethazine-d3 (hydrochloride) (CRM) (Cay-39606) is intended for use as an internal standard for the quantification of promethazine (Cay-21331, Cay-22450) by GC- or LC-MS. Promethazine is categorized as a phenothiazine. It has been associated with misuse in conjunction with opioids or sedatives. Formulations...
| Keywords: | N,alpha-dimethyl-N-(methyl-d3)-10H-phenothiazine-10-ethanamine, monohydrochloride |
| Application: | GC-MS, LC-MS, internal standard, quantification, phenothiazine, Histamine receptor H1 antagonist |
| CAS | 1435933-86-0 |
| MW: | 323.9 D |
172.00€
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Levocetirizine
Item number: TGM-T1469-100mg
Description: Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist. Target: Histamine Receptor. Smiles: [C@H](N1CCN(CCOCC(O)=O)CC1)(C2=CC=C(Cl)C=C2)C3=CC=CC=C3. References: Pasquali M, et al. Clin Exp Allergy. 2006 Sep,36(9):1161-7.
| Keywords: | Levocetirizine HCl |
| Application: | Targets histamine receptor H1 (HRH1) |
| CAS | 130018-77-8 |
| MW: | 388.89 D |
From 33.00€
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Fexofenadine hydrochloride
Item number: TGM-T1470-10mg
Description: Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis, angioedema and chronic urticaria. Target: Histamine Receptor. Smiles: Cl.CC(C)(C(O)=O)c1ccc(cc1)C(O)CCCN1CCC(CC1)C(O)(c1ccccc1)c1ccccc1....
| Keywords: | Terfenidine carboxylate hydrochloride, MDL-16455 hydrochloride, Telfast, MDL 16455A, Allegra, Fexofenadine HCl |
| Application: | Targets histamine receptor H1 (HRH1) |
| CAS | 153439-40-8 |
| MW: | 538.13 D |
From 45.00€
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Carbinoxamine
Item number: TGM-T21247-25mg
Description: Carbinoxamine, an anticholinergic and antihistamine agent, is used for hay fever, angioedema, vasomotor rhinitis, mild urticaria, dermatographism and allergic conjunctivitis. It is a histamine antagonist, specifically an H1-antagonist. Target: Others. Smiles: C(OCCN(C)C)(C1=CC=C(Cl)C=C1)C2=CC=CC=N2....
| Keywords: | Paracarbinoxamine, (+-)-Carbinoxamine, Allergefon |
| Application: | Targets histamine receptor H1 (HRH1) |
| CAS | 486-16-8 |
| MW: | 290.79 D |
From 1,491.00€
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Dimethindene maleate
Item number: TGM-T21472-1mg
Description: Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis. Target: Histamine Receptor. Smiles: OC(=O)\C=C/C(O)=O.CC(C1=C(CCN(C)C)Cc2ccccc12)c1ccccn1. References: Towart R, et al. Investigation of the...
| Keywords: | SU 6518, UNII-6LL60J9E0O, SU-6518 |
| Application: | Targets histamine receptor H1 (HRH1) |
| CAS | 3614-69-5 |
| MW: | 408.49 D |
From 41.00€
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Quifenadine
Item number: TGM-T20951-25mg
Description: Quifenadine, an H1-histamine receptor blocker, has antiarrhythmic properties. Target: Others. Smiles: OC(C1CN2CCC1CC2)(C1=CC=CC=C1)C1=CC=CC=C1. References: Luss LV. [Use of antihistamines in a physician's clinical practice]. Ter Arkh. 2014,86(8):106-9. Review. Russian. PubMed PMID: 25306755.
| Keywords: | Phencarol, Fenatin, Fencarol |
| Application: | Targets histamine receptor H1 (HRH1) |
| CAS | 10447-39-9 |
| MW: | 293.4 D |
From 1,491.00€
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Thonzylamine hydrochloride
Item number: TGM-T21014-5mg
Description: Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic. Target: Histamine Receptor, AChR. Smiles: Cl.N=1C=CC=NC1N(CC2=CC=C(OC)C=C2)CCN(C)C. References: Sabry SM, et al. Sensitive spectrofluorimetric and spectrophotometric methods for the determination of...
| Keywords: | Resistab, Thonzylamine HCl, Novohetramin, Neohetramine hydrochloride, Anahist |
| Application: | Targets histamine receptor H1 (HRH1) |
| CAS | 63-56-9 |
| MW: | 322.83 D |
From 50.00€
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Antazoline phosphate
Item number: TGM-T21020-500mg
Description: Antazoline phosphate is an antihistamine with anticholinergic properties. Antazoline prevents the typical allergic symptoms on capillaries, mucous membranes, skin, and gastrointestinal and bronchial smooth muscles by antagonizing the histamine H1 receptor. Target: Others. Smiles:...
| Application: | Targets histamine receptor H1 (HRH1) |
| CAS | 154-68-7 |
| MW: | 363.35 D |
1,342.00€
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Emedastine Difumarate
Item number: TGM-T21388-5mg
Description: Emedastine Difumarate is a selective histamine H1 receptor antagonist with anti-allergic activity, prescribed for allergic conjunctivitis. Upon ocular administration, emedastine causes a dose-dependent inhibition of histamine-stimulated vascular permeability in the conjunctiva. Target: Others. Smiles:...
| Keywords: | DSSTox_CID_26911, Rapimine, AL-3432A, KB-2413, Emedastine fumarate, KB 2413 |
| Application: | Targets histamine receptor H1 (HRH1) |
| CAS | 87233-62-3 |
| MW: | 534.56 D |
951.00€
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Mianserin
Item number: TGM-T21428-1mg
Description: Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific...
| Keywords: | Norval, Lantanon, Lumin, Depnon, Lerivon |
| Application: | Targets 5-hydroxytryptamine receptor 2 (HTR2) |
| CAS | 24219-97-4 |
| MW: | 264.36 D |
From 388.00€
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Olopatadine
Item number: TGM-T21462-25mg
Description: Olopatadine, an antihistamine, as well as anticholinergic and mast cell stabilizer, is used for the treatment of itching associated with allergic conjunctivitis (eye allergies). There is also a potential for Olopatadine to treat steroid rebound (red skin syndrome). Target: Others. Smiles:...
| Keywords: | KW-4679, KW-4943A, Opatanol, Patanol |
| Application: | Targets histamine receptor H1 (HRH1) |
| CAS | 113806-05-6 |
| MW: | 337.41 D |
1,491.00€
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