223 products were found matching "K04145"!
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Tiapride hydrochloride
Item number: TGM-T1292-50mg
Description: Tiapride is a selective blocker of D2/3 dopamine receptors in the brain. It is used in the therapy of various psychiatric and neurological disorders containing dyskinesia, negative symptoms of psychosis, alcohol withdrawal syndrome, and aggression and agitation in the elderly. Target: Dopamine Receptor....
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 51012-33-0 |
| MW: | 364.89 D |
36.00€
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Ziprasidone D8
Item number: TGM-T13400-10mg
Description: Ziprasidone D8 is deuterium labeled Ziprasidone, which is a antagonist of combined 5-HT (serotonin) and dopamine receptor and exhibits potent effects of antipsychotic activity. Smiles: [2H]C1([2H])N(CCc2cc3CC(=O)Nc3cc2Cl)C([2H])([2H])C([2H])([2H])N(c2nsc3ccccc23)C1([2H])[2H]
| Keywords: | CP-88059 D8 |
| Application: | GC-MS, LC-MS, internal standard, dopamine D2-receptor antagonist |
| CAS | 1126745-58-1 |
| MW: | 420.99 D |
From 576.00€
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Loxapine succinate
Item number: TGM-T1412-100mg
Description: Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia. Target: Dopamine Receptor, 5-HT Receptor. Smiles: OC(=O)CCC(=O)O.CN1CCN(CC1)C1=Nc2ccccc2Oc2c1cc(Cl)cc2. References: Singh AN, et al. J Psychiatry Neurosci, 1996, 21(1), 29-35.
| Keywords: | Loxapine succinate salt, Daxolin, Cloxazepin, Loxapac |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 27833-64-3 |
| MW: | 445.9 D |
From 33.00€
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Trifluoperazine dihydrochloride
Item number: TGM-T1222-100mg
Description: Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic. Target: CaMK, Adrenergic Receptor, Autophagy, P-gp, Dopamine Receptor, Influenza Virus. Smiles: Cl.CN1CCN(CCCN2C3=CC=CC=C3SC3=C2C=C(C=C3)C(F)(F)F)CC1. References: Lahti...
| Keywords: | Trifluoperazine 2HCl, SKF5019, Urinox |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 440-17-5 |
| MW: | 480.43 D |
50.00€
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Risperidone E-oxime
Item number: TGM-T12734-1mg
Description: Risperidone E-oxime is an impurity of Risperidone, a serotonin 5-HT2 receptor blocker, P-glycoprotein inhibitor, and potent dopamine D2 receptor antagonist (Kis of 4.8 and 5.9 nM for 5-HT2A and dopamine D2 receptors, respectively). Target: Others. Smiles:...
| Application: | Potential impurity |
| CAS | 691007-09-7 |
| MW: | 430.49 D |
281.00€
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Pimozide-d4
Item number: TGM-T12476-10mg
Description: Pimozide D4 is a deuterium labeled Pimozide. Smiles: O=C1N(C=2C(N1)=CC=CC2)C3CCN(CCCC(C4=C(C(=C(F)C(=C4[2H])[2H])[2H])[2H])C5=CC=C(F)C=C5)CC3. References: Ybema CE, et al. Adrenoceptors and dopamine receptors are not involved in the discriminative stimulus effect of the 5-HT1A receptor agonist...
| Keywords: | R6238 D4, Pimozide D4 |
| Application: | GC-MS, LC-MS, internal standard, quantification, dopamine D2/D3-receptor antagonist |
| CAS | 1803193-57-8 |
| MW: | 465.57 D |
From 909.00€
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Bromperidol
Item number: TGM-T14830-10mg
Description: Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic. Which is used as an antipsychotic in the treatment of schizophrenia. Target: 5-HT Receptor. Smiles: OC1(CCN(CCCC(=O)c2ccc(F)cc2)CC1)c1ccc(Br)cc1. References: Marianna Purgato, Clive E Adams.Bromperidol...
| Keywords: | R-11333 |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 10457-90-6 |
| MW: | 420.32 D |
From 31.00€
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Cabergoline
Item number: TGM-T14853-100mg
Description: Cabergoline (FCE-21336) is an ergot derived-dopamine D2-like receptor agonist. It has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively).Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels....
| Keywords: | FCE-21336 |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 81409-90-7 |
| MW: | 451.6 D |
From 34.00€
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Talipexole dihydrochloride
Item number: TGM-T14490-100mg
Description: Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, alpha2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and intestinal membrane fractions with Ki values of 0.35 µM and 0.22 µM, respectively. It displays antiParkinsonian activity. Target: Adrenergic...
| Keywords: | Domnin, B-HT 920 dihydrochloride |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 36085-73-1 |
| MW: | 282.23 D |
From 33.00€
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Pramipexole
Item number: TGM-T1476-1mL
Description: Pramipexole (SND 919) is a selective dopamine receptor agonist used in the therapy of Parkinson disease. Pramipexole therapy is associated with a low rate of transient serum enzyme elevations during treatment but has not been implicated in cases of clinically apparent acute liver injury. Target:...
| Keywords: | SND 919 |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 104632-26-0 |
| MW: | 211.33 D |
From 42.00€
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Brilaroxazine
Item number: TGM-T14782-100mg
Description: Brilaroxazine (RP5063) is a potent multimodal dopamine/5-HT modulator. Brilaroxazine is a partial agonist of dopamine D2, D3, and D4 receptors, 5-HT1A (Ki =1.5 nM) and 5-HT2A (Ki = 2.5 nM), and has antagonist activity 5-HT2B, and 5-HT7 receptors with Kis of 0.19 nM and 2.7 nM, respectively....
| Keywords: | RP5063 |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 1239729-06-6 |
| MW: | 450.36 D |
From 105.00€
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Aripiprazole Lauroxil
Item number: TGM-T14319-100mg
Description: Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic. Aripiprazole lauroxil is cleaved by esterases in vivo to N-hydroxymethyl aripiprazole (lauric acid), which is then cleaved to aripiprazole, which is non-toxic. Target: 5-HT Receptor,...
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 1259305-29-7 |
| MW: | 660.71 D |
From 41.00€
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