79 products were found matching "K04144"!
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DRD1 Reporter Assay System (human)
Item number: IB-IB46001
This is an all-inclusive cell-based luciferase reporter assay kit targeting the the Human Dopamine Receptor D1 (DRD1). INDIGO's DRD1 reporter assay utilizes proprietary mammalian cells that have been engineered to provide constitutive expression of the DRD1. In addition to DRD1 Reporter Cells, this kit provides two...
| Keywords: | DRD1, Dopamine D1 receptor, D(1A) dopamine receptor |
| Application: | Functional activity screening |
| Species reactivity: | human |
From 1,507.00€
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Pergolide
Item number: TGM-T21340-25mg
Description: Pergolide, an ergoline-based dopamine receptor agonist, is used for the treatment of Parkinson's disease, which is associated with low levels of the neurotransmitter dopamine in the brain. Target: Others. Smiles: CCCN1C[C@H](CSC)CC2[C@H]1Cc1c[nH]c3cccc2c13
| Application: | Targets dopamine receptor D1 (DRD1) |
| CAS | 66104-22-1 |
| MW: | 314.49 D |
From 1,520.00€
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A 77636 hydrochloride
Item number: TGM-T21782-1mg
Description: A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40, Ki=39.8 nM). A 77636 hydrochloride shows antiparkinsonian activity. A 77636 hydrochloride is functionally inactive at dopamine D2 receptor. Target: Dopamine Receptor. Smiles:...
| Keywords: | A77636 hydrochloride |
| Application: | Dopamine D1 receptor agonist |
| CAS | 145307-34-2 |
| MW: | 365.89 D |
From 97.00€
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Flupenthixol
Item number: TGM-T21401-25mg
Description: Flupentixol is a typical antipsychotic drug of the thioxanthene class. Flupentixol is also used in low doses as an antidepressant. Target: Others. Smiles: C(CCN1CCN(CCO)CC1)=C2C=3C(SC=4C2=CC=CC4)=CC=C(C(F)(F)F)C3. References: Tardy M, Dold M, Engel RR, Leucht S. Flupenthixol versus low-potency...
| Keywords: | Emergil, Fluanxol, Siplaril, Depixol |
| Application: | Targets dopamine receptor D1 (DRD1) |
| CAS | 2709-56-0 |
| MW: | 434.52 D |
From 1,520.00€
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Zicronapine
Item number: TGM-T35307-100mg
Description: Zicronapine( LU 31-130) is an atypical antipsychotic. Zicronapine has monoaminergic activity and multi-receptor properties. It has shown effective antagonism against dopamine D1, D2, and serotonin 5HT2A receptors in vitro and in vivo. Target: Others. Smiles:...
| Keywords: | Lu-31130, Lu31-130, Lu 31-130, Lu 31130, Lu31130, Lu-31-130 |
| Application: | Targets 5-hydroxytryptamine receptor 2 (HTR2) |
| CAS | 170381-16-5 |
| MW: | 354.92 D |
From 1,520.00€
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Adrogolide HCl
Item number: TGM-T29674-25mg
Description: Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist. Target: Others. Smiles: O(C(C)=O)C=1C=C2[C@]3(C4=C(SC(CCC)=C4)CN[C@@]3(CCC2=CC1OC(C)=O)[H])[H].Cl. References: Gleason SD, Witkin JM. Effects of dopamine D1 receptor full agonists in rats trained to discriminate SKF 38393. Behav...
| Keywords: | DAS 431, ABT 431, A-93431.1, ABT 431,ABT-431,ABT431, ABT431, Adrogolide Hydrochloride, ABT-431 |
| Application: | Targets dopamine receptor D1 (DRD1) |
| CAS | 166591-11-3 |
| MW: | 435.96 D |
From 2,272.00€
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Pipotiazine
Item number: TGM-T34072-100mg
Description: Pipotiazine has less sedating and a weak propensity for causing hypotension or potentiating the effects of CNS depressants and anesthetics among the different phenothiazine derivatives. However, it produces a high incidence of extra pyramidal reactions. It is used for the maintenance treatment of...
| Keywords: | Pipothiazine, Piportil L4, Pipotiazinum, Pipotiazina, 19366 RP |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 39860-99-6 |
| MW: | 475.67 D |
From 1,520.00€
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Carphenazine Dimaleate
Item number: TGM-T30753-100mg
Description: Carphenazine is used for the treatment of chronic schizophrenia, which is an antipsychotic agent. Target: Others. Smiles: OC(=O)\C=C/C(O)=O.OC(=O)\C=C/C(O)=O.CCC(=O)c1ccc2Sc3ccccc3N(CCCN3CCN(CCO)CC3)c2c1. References: MILLER G. EVALUATION OF TWO TRANQUILIZERS: ACETOPHENAZINE MALEATE (TINDAL MALEATE):...
| Keywords: | carphenazine maleate, Proketazine, Proketazine maleate, Procethazine dimaleate, Proketazine dimaleate |
| Application: | Targets dopamine receptor D1 (DRD1) |
| CAS | 2975-34-0 |
| MW: | 657.74 D |
From 1,520.00€
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Zuclopenthixol
Item number: TGM-T4117-100mg
Description: Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors. Target: Dopamine Receptor. Smiles: OCCN1CCN(CC\C=C2\c3ccccc3Sc3ccc(Cl)cc23)CC1. References: Khalifa AE: Zuclopenthixol...
| Keywords: | (Z)-Clopenthixol, Cisordinol, cis-Clopenthixol |
| Application: | Targets dopamine receptor D1 (DRD1) |
| CAS | 53772-83-1 |
| MW: | 400.96 D |
From 30.00€
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Zuclopenthixol decanoate
Item number: TGM-T4117L-100mg
Description: Zuclopenthixol decanoate is an anti-schizophrenia drug. Target: Others. Smiles: C(\CCN1CCN(CCOC(CCCCCCCCC)=O)CC1)=C/2\C=3C(SC=4C2=CC=CC4)=CC=C(Cl)C3. References: Cordiner M, Shajahan P, McAvoy S, Bashir M, Taylor M. Effectiveness of long-acting antipsychotics in clinical practice : 1. A retrospective,...
| Keywords: | Zuclopenthixol, Zuclopenthixol HCl |
| Application: | Targets dopamine receptor D1 (DRD1) |
| CAS | 64053-00-5 |
| MW: | 555.21 D |
From 1,520.00€
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SCH-23390 hydrochloride
Item number: TGM-T4369-100mg
Description: SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, with high affinity for the D1 (Ki=0.2 nM) and D5 (Ki=0.3 nM) receptors. Target: 5-HT Receptor, Dopamine Receptor, Potassium Channel. Smiles: Cl.CN1CCc2cc(Cl)c(O)cc2[C@H](C1)c1ccccc1. References: Bourne...
| Keywords: | R-(+)-SCH23390 hydrochloride |
| Application: | Dopamine receptor D1 / D5 antagonist |
| CAS | 125941-87-9 |
| MW: | 324.24 D |
From 34.00€
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Flupentixol dihydrochloride
Item number: TGM-T5135-100mg
Description: Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders. Target: Dopamine Receptor. Smiles: OCCN1CCN(CC1)CCC=C2c3c(Sc4c2cc(C(F)(F)F)cc4)cccc3.Cl.Cl. References: Yonar D, et al. Effect of cis-(Z)-flupentixol on DPPC membranes in the presence and...
| Keywords: | (E/Z)-Flupentixol Dihydrochloride, Flupenthixol dihydrochloride, Fupentixol Dihydrochloride |
| Application: | Targets dopamine receptor D1 (DRD1) |
| CAS | 2413-38-9 |
| MW: | 507.43 D |
From 40.00€
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