105 products were found matching "K04141"!

Organism: Mus musculus (Mouse). Source: in vitro E.coli expression system. Expression Region: 1-466aa. Protein Length: Full Length. Tag Info: N-terminal 6xHis-SUMO-tagged. Target Protein Sequence: MGAGALALGA SEPCNLSSAA PLPDGAATAA RLLVLASPPA SLLPPASEGS APLSQQWTAG MGLLLALIVL LIVVGNVLVI VAIAKTPRLQ TLTNLFIMSL ASADLVMGLL...

CGP 20712A is an antagonist of the beta1-adrenergic receptor (beta1-AR, IC50 = 0.7 nM). It is selective for beta1-ARs over beta2-ARs (IC50 = 6,700 nM). CGP 20712 A (0.1-1,000 µM) inhibits adenylyl cyclase activity induced by the beta1- and beta2-AR agonist isoproterenol (Cay-15592) in brown adipose tissue plasma...

This is an all-inclusive cell-based luciferase reporter assay kit targeting the the Human Adrenoreceptor Beta 1 (ADRB1). INDIGO's ADRB1 reporter assay utilizes proprietary mammalian cells that have been engineered to provide constitutive expression of the ADRB1. In addition to ADRB1 Reporter Cells, this kit provides...

This is an all-inclusive cell-based luciferase reporter assay kit targeting the the Human Adrenoreceptor Beta 1 (ADRB1). INDIGO's ADRB1 reporter assay utilizes proprietary mammalian cells that have been engineered to provide constitutive expression of the ADRB1. In addition to ADRB1 Reporter Cells, this kit provides...

Betaxolol-d7 is intended for use as an internal standard for the quantification of betaxolol (Cay-18625) by GC- or LC-MS. Betaxolol is an antagonist of the beta1-adrenergic receptor (beta1-AR, Ki = 23 nM). It is selective for the beta1-AR over the beta2-AR (Ki = 790 nM). Betaxolol is cytotoxic to 10.014 pRSV-T human...

The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Mouse ADRb1. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Mouse ADRb1. Next,...

The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human ADRb1. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Human ADRb1. Next,...

The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Rat ADRb1. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Rat ADRb1. Next,...

A b-Adrenergic receptor selective antagonist used as a antiglaucoma agent.

(±)-Talinolol is a beta1-selective adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity. By blocking beta1-adrenergic receptors, talinolol delays the conduction of stimuli in the AV node, reduces the sino-atrial conduction time, and impedes the sinus node automaticity. Because...

Isoproterenol is an agonist of beta1- and beta2-adrenergic receptors (beta1- and beta2-ARs, Kis = 224 and 458 nM, respectively. It is selective for beta1- and beta2-ARs over beta3-ARs (Ki = 1,570 nM). Isoproterenol inhibits contractions in isolated field-stimulated rat vas deferens (EC50 = 45.6 nM). In vivo,...

Metoprolol tartrate is a beta1-adrenergic blocker.