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GSK-5959
Item number: TGM-T1972-100mg
Description: GSK-5959 is an effective, specific and cell permeable BRPF1 bromodomain inhibitor (IC50: ~80 nM). The selectivity of GSK-5959 for BRPF1 is >100-fold over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Target: Epigenetic Reader Domain. Smiles:...
| Application: | BRPF1 (Peregrin) bromodomain inhibitor |
| CAS | 901245-65-6 |
| MW: | 394.47 D |
From 52.00€
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GSK5959
Item number: Cay18123-5
The bromodomain and PHD finger-containing (BRPF) proteins are scaffolding components of chromatin-binding MOZ/MORF histone acetyltransferase complexes, which have activity as transcriptional regulators. BRPF1 (BR140 or Peregrin) is important for maintaining Hox gene expression and the development of multiple...
| Keywords: | N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxy-benzamide |
| Application: | Cell-permeable BRPF1 bromodomain inhibitor |
| CAS | 901245-65-6 |
| MW: | 394.5 D |
From 44.00€
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GSK-5959
Item number: BPS-82066
GSK-5959 exhibits >100-fold selectivity for BRPF1 (IC50 = 80 nM) over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3, which is involved in the epigenetic regulation of gene expression and have been implicated in human cancer.
| Keywords: | GSK5959, GSK 5959, |
| Application: | BRPF1 (Peregrin) bromodomain inhibitor |
| CAS | 901245-65-6 |
| MW: | 394,5 D |
710.00€
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