2 products were found matching "870653-45-5"!

No results were found for the filter!
PAP-1
PAP-1

Item number: TGM-TQ0179-100mg

Description: PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, orally active Kv1.3 blocker with an EC50 of 2 nM. Target: Potassium Channel. Smiles: O=c1ccc2c(OCCCCOc3ccccc3)c3ccoc3cc2o1. References: Schmitz A, et al. Design of PAP-1, a selective small molecule Kv1.3 blocker, for the suppression of effector memory...
Keywords: 5-(4-Phenoxybutoxy)psoralen
Application: Kv1.3 channels inhibitor
CAS 870653-45-5
MW: 350.36 D
From 57.00€ *
Review
PAP-1
PAP-1

Item number: Cay30105-1

PAP-1 is an inhibitor of Kv1.3 voltage-gated potassium channels (EC50 = 2 nM at -80 mV in cells overexpressing the human channel). It is selective for Kv1.3 over a panel of 22 ion channels, including potassium, sodium, calcium, and chloride channels (EC50s = 45-15,000 nM for all). PAP-1 inhibits anti-CD3...
Keywords: 5-(4-Phenoxybutoxy)psoralen, 4-(4-phenoxybutoxy)-7H-furo[3,2-g][1]benzopyran-7-one
Application: Kv1.3 channels inhibitor
CAS 870653-45-5
MW: 350.4 D
From 55.00€ *
Review