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BPTU
Item number: TGM-T4132-100mg
Description: BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 µM). Non-nucleotide ligand. Binds receptor outside of the helical bundle. Blocks inhibition of spontaneous contraction of rat and mouse colon induced by electrical field stimulation, nicotine and P2Y agonists. Antithrombotic, reduces...
| Keywords: | BMS-646786 |
| Application: | Allosteric P2Y1 receptor antagonist |
| CAS | 870544-59-5 |
| MW: | 445.43 D |
From 33.00€
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BPTU
Item number: Cay29444-10
BPTU is an allosteric antagonist of the purinergic P2Y1 receptor (Ki = 6 nM for the human receptor). BPTU is selective for P2Y1 over P2Y2, P2Y6, P2Y11, P2Y12, and P2Y14 receptors (Kis = >3,500 nM). It inhibits platelet aggregation in human platelet-rich plasma (hPRP, IC50 = 2.1 µM). BPTU reduces thrombus weight by...
| Keywords: | N-[2-[2-(1,1-dimethylethyl)phenoxy]-3-pyridinyl]-N'-[4-(trifluoromethoxy)phenyl]-urea |
| Application: | Allosteric P2Y1 receptor antagonist |
| CAS | 870544-59-5 |
| MW: | 445.4 D |
From 44.00€
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