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Esmolol hydrochloride
Esmolol hydrochloride

Item number: TGM-T1503-1mL

Description: Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instances of clinically apparent drug induced liver injury. Target: Mitophagy, Adrenergic Receptor, Autophagy. Smiles:...
Keywords: ASL8052, Esmolol HCl
Application: Targets adrenergic receptor beta-1 (ADRB1)
CAS 81161-17-3
MW: 331.15 D
From 50.00€ *
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Esmolol (hydrochloride)
Esmolol (hydrochloride)

Item number: Cay22581-10

Esmolol is a beta1-adrenergic receptor (beta1-AR) antagonist. It binds to beta1-ARs (Kd = 100 nM in isolated cardiac myocytes) and is 34-fold selective for beta1- over beta2-ARs. Esmolol also inhibits L-type Ca2+ currents (ICa.L) and the fast Na+ current (INa) in rat cardiac myocytes (IC50s = 50 and 169 µM,...
Keywords: ASL 8052, 4-[2-hydroxy-3-[(1-methylethyl)amino]propoxy]-benzenepropanoic acid, methyl ester, monohydrochloride
Application: beta1-Adrenergic receptor antagonist
CAS 81161-17-3
MW: 331.8 D
From 43.00€ *
Review