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GS-6201
Item number: TGM-T15418-100mg
Description: GS-6201 (CVT-6883) is a selective antagonist of the adenosine A2B receptor, demonstrating high affinity and selectivity with a Ki of 22 nM for human adenosine A2B receptors. Target: Adenosine Receptor. Smiles: CCCn1c(=O)n(CC)c2[nH]c(nc2c1=O)-c1cnn(Cc2cccc(c2)C(F)(F)F)c1. References: Toldo S, et al....
| Keywords: | CVT-6883 |
| Application: | Adenosine A2B receptor antagonist |
| CAS | 752222-83-6 |
| MW: | 446.43 D |
From 38.00€
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CVT-6883
Item number: Cay33333-1
CVT-6883 is an adenosine A2B receptor antagonist (Ki = 22 nM). It is selective for adenosine A2B over adenosine A1, A2A, and A3 receptors (Kis = 1,940, 3,280, and 1,070 nM, respectively), as well as a panel of 84 receptors, ion channels, transporters, and enzymes at 10 µM. CVT-6883 (6 mg/kg) decreases allergen...
| Keywords: | GS-6201, 3-ethyl-3,9-dihydro-1-propyl-8-[1-[[3-(trifluoromethyl)phenyl]methyl]-1H-pyrazol-4-yl]-1H-purine-2,6-dione |
| Application: | Adenosine A2B receptor antagonist |
| CAS | 752222-83-6 |
| MW: | 446.4 D |
From 44.00€
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