2 products were found matching "737789-87-6"!

No results were found for the filter!
Relugolix
Relugolix

Item number: TGM-T3630-100mg

Description: Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential antineoplastic activity. Relugolix competitively binds to and blocks the GnRH receptor in the anterior pituitary gland, which both...
Keywords: RVT-601, TAK-385
Application: Targets gonadotropin-releasing hormone receptor (GNRHR)
CAS 737789-87-6
MW: 623.63 D
From 32.00€ *
Review
TAK-385
TAK-385

Item number: Cay29512-1

TAK-385 is an orally bioavailable gonadotropin-releasing hormone receptor (GnRHR) antagonist (IC50s = 0.33 and 0.32 nM for the human and monkey receptors, respectively). It is selective for these receptors over the rat GnRHR receptor (IC50 = 9,800 nM), as well as a panel of 134 enzymes and receptors at 10 µM....
Keywords: Relugolix,...
Application: GnRHR antagonist
CAS 737789-87-6
MW: 623.6 D
From 43.00€ *
Review