2 products were found matching "681806-46-2"!

No results were found for the filter!
BRL 44408 Maleate Salt
BRL 44408 Maleate Salt

Item number: TGM-T26904-10mg

Description: BRL 44408 Maleate Salt is a selective alpha2A-adrenoceptor antagonist with Ki value of 1.7 nM. BRL 44408 Maleate Salt increases the release of hippocampal noradrenalin following systemic administration. Target: Others. Smiles: C(=C\C(O)=O)\C(O)=O.CC1C=2C(CN1CC=3NCCN3)=CC=CC2. References: Dwyer JM, Platt...
Keywords: BRL 44408, BRL-44408, BRL44408
CAS 681806-46-2
MW: 331.37 D
From 210.00€ *
Review
BRL 44408 (maleate)
BRL 44408 (maleate)

Item number: Cay29454-10

BRL 44408 is an antagonist of alpha2A-adrenergic receptors (alpha2A-ARs, Ki = 8.56 nM for the recombinant human receptors). It is greater than 50-fold selective for alpha2A-ARs over alpha1-, alpha2B-, alpha2C-, beta1-, and beta2-ARs, as well as 19 other neurotransmitter receptors, transporters, and enzymes in a...
Keywords: 2-[(4,5-dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole, 2Z-butenedioate
Application: alpha2A-adrenergic receptor antagonist
CAS 681806-46-2
MW: 331.4 D
From 115.00€ *
Review