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Droperidol
Item number: TGM-T0990-100mg
Description: Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist. Target: Dopamine Receptor. Smiles: O=C1N(C=2C(N1)=CC=CC2)C=3CCN(CCCC(=O)C4=CC=C(F)C=C4)CC3. References: Kao LW, et al. Ann Emerg Med, 2003, 41(4), 546-558.
| Keywords: | Dehydrobenzperidol, NSC 169874 |
| CAS | 548-73-2 |
| MW: | 379.43 D |
From 40.00€
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Droperidol
Item number: Cay18884-1
Droperidol is a dopamine D2 and D4 receptor antagonist (Kis = 0.25 and 0.84 nM for human D2 and D4 receptors, respectively). It also inhibits the voltage-gated potassium channel hERG, also known as Kv11.1 (IC50 = 32 nM), and binds to the serotonin (5-HT) receptor subtype 5-HT2 (Ki = 1.1 nM). Droperidol (1, 5, and 10...
| Keywords: | NSC 169874, 1-[1-[4-(4-fluorophenyl)-4-oxobutyl]-1,2,3,6-tetrahydro-4-pyridinyl]-1,3-dihydro-2H-benzimidazol-2-one |
| Application: | Dopamine D2-receptor antagonist |
| CAS | 548-73-2 |
| MW: | 379.4 D |
From 44.00€
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Droperidol
Item number: CDX-D0823-G001
White to light yellow powder. Soluble in DMSO (20mg/ml) or DMF (20mg/ml). Chemical. CAS: 548-73-2. Formula: C22H22FN3O2. MW: 379.43. Droperidol is a butyrophenone that acts as an antagonist at dopamine receptors D2 and D4. It less potently inhibits the human voltage-gated potassium channel, 5-HT, alpha-adrenergic...
| Keywords: | 1-[1-[3-(p-Fluorobenzoyl)propyl]-1,2,3,6-tetrahydro-4-pyridyl]-2-benzimidazolinone, NSC 169874 |
| CAS | 548-73-2 |
| MW: | 379,43 D |
From 122.00€
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