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Preladenant
Item number: TGM-T4290-100mg
Description: Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine receptors. Target: Adenosine Receptor. Smiles: COCCOc1ccc(cc1)N1CCN(CCn2ncc3c2nc(N)n2nc(nc32)-c2ccco2)CC1. References: Hodgson RA, et al....
| Keywords: | SCH-420814 |
| Application: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| CAS | 377727-87-2 |
| MW: | 503.56 D |
From 31.00€
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Preladenant
Item number: Cay22210-1
Preladenant is an orally bioavailable antagonist of the adenosine A2A receptor (Kis = 1.1 and 2.5 nM for human and rat receptors, respectively). It is selective for A2A receptors over A1, A2B, and A3 receptors (Kis = >1,000, >1,700, and >1,000 nM, respectively) as well as a panel of 59 receptors, enzymes, and ion...
| Keywords: | SCH 420814,... |
| Application: | Adenosine receptor A2a antagonist |
| CAS | 377727-87-2 |
| MW: | 503.6 D |
From 35.00€
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