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JTC-801
Item number: TGM-T6553-10mg
Description: JTC-801 is a selective opioid receptor-like 1 (ORL1) receptor antagonist with an IC50 of 94 nM and weak inhibitory effects on delta, kappa, and µ receptors. Target: Opioid Receptor. Smiles: Cl.CCc1ccc(OCc2ccccc2C(=O)Nc2ccc3nc(C)cc(N)c3c2)cc1. References: Yamada H, et al. Br J Pharmacol, 2002, 135(2),...
| Keywords: | JTC 801, JTC801 |
| Application: | ORL1 antagonist |
| CAS | 244218-51-7 |
| MW: | 447.96 D |
From 41.00€
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JTC 801
Item number: Cay21254-5
JTC 801 is an antagonist of the nociceptin receptor (ORL1, Ki = 44.5 nM, IC50 = 94 nM) that is >100-, >100-, and >3-fold more selective for ORL1 over the related delta-, kappa-, and µ-opioid receptors, respectively. It demonstrates anti-nociceptive effects in acute pain models in mice upon oral administration at 1...
| Keywords: | N-(4-amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]-benzamide, monohydrochloride |
| Application: | ORL1 antagonist |
| CAS | 244218-51-7 |
| MW: | 448 D |
From 77.00€
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