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Masofaniten
Masofaniten

Item number: Cay41670-1

Masofaniten is an androgen receptor N-terminal transactivation domain inhibitor (ARTADI). It binds to the tryptophan residues in positions 397 (W397) and W433 in the AR TAD.Formal Name: N-[4-[[4-[1-[3-chloro-4-(2-chloroethoxy)-5-cyanophenyl]-1-methylethyl]phenoxy]methyl]-2-pyrimidinyl]-methanesulfonamide. CAS...
Keywords: EPI-7386,...
Application: Androgen receptor N-terminal transactivation domain inhibitor (ARTADI)
CAS 2416716-62-4
MW: 535.4 D
From 146.00€ *
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Masofaniten
Masofaniten

Item number: TGM-T72985-100mg

Description: Masofaniten (Androgen receptor-IN-2), a potent, orally active inhibitor of the androgen receptor, demonstrates significant antitumor activity against prostate cancer. Target: Others. Smiles: C(C)(C)(C1=CC(C#N)=C(OCCCl)C(Cl)=C1)C2=CC=C(OCC3=NC(NS(C)(=O)=O)=NC=C3)C=C2
Keywords: Androgen receptor-IN-2
Application: Targets androgen receptor (AR, NR3C4)
CAS 2416716-62-4
MW: 535.44 D
From 1,620.00€ *
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