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LSZ-102
Item number: Cay41834-1
LSZ-102 is an estrogen receptor alpha (ERalpha) degrader (IC50 = 0.2 nM). It reduces 17beta-estradiol-induced transcription in a reporter assay using MCF-7 breast cancer cells expressing ERalpha (IC50 = 6 nM). LSZ-102 decreases the proliferation of MCF-7 cells (IC50 = 1.7 nM). In vivo, LSZ-102 (20 mg/kg per day)...
| Keywords: | 3-[4-[[2E-[2-(1,1-difluoroethyl)-4-fluorophenyl]-6-hydroxybenzo[b]thien-3-yl]oxy]phenyl]-2-propenoic acid |
| Application: | ERalpha degrader |
| CAS | 2135600-76-7 |
| MW: | 470.5 D |
From 62.00€
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LSZ-102
Item number: TGM-T15788-10mg
Description: LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERalpha positive breast cancer. Target: Estrogen Receptor/ERR. Smiles: CC(F)(F)c1cc(F)ccc1-c1sc2cc(O)ccc2c1Oc1ccc(\C=C\C(O)=O)cc1. References: Tria GS, et al. Discovery of LSZ102, a...
| Keywords: | LSZ102 |
| CAS | 2135600-76-7 |
| MW: | 470.46 D |
From 79.00€
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