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Item number: Cay24480-10

SR 17018 is an orally bioavailable and brain-penetrant agonist of µ-opioid receptors. It is functionally selective for G protein-coupled receptor signaling (EC50 = 97 nM for GTPgammaS binding in CHO cells expressing µ-opioid receptors) over beta-arrestin 2 recruitment (EC50 = >10,000 nM) at the µ-opioid receptor. SR...

Keywords:	5,6-dichloro-1-[1-[(4-chlorophenyl)methyl]-4-piperidinyl]-1,3-dihydro-2H-benzimidazol-2-one
Application:	µ-opioid receptor agonist
CAS	2134602-45-0
MW:	410.7 D

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SR17018

Item number: TGM-T4407-100mg

Description: SR17018, a mu-opioid receptor (MOR) agonist, binds with GTPgammaS and has an EC50 of 97 nM. Target: Opioid Receptor. Smiles: Clc1ccc(CN2CCC(CC2)n2c3cc(Cl)c(Cl)cc3[nH]c2=O)cc1. References: Schmid CL,etal.Bias Factor and Therapeutic Window Correlate to Predict Safer Opioid Analgesics.Cell. 2017 Nov...

Application:	µ-opioid receptor agonist
CAS	2134602-45-0
MW:	410.72 D

From 63.00€ *

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