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Methiothepin maleate
Item number: TGM-T4375-100mg
Description: Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors. Target: 5-HT Receptor. Smiles: OC(=O)\C=C/C(O)=O.CSc1ccc2Sc3ccccc3CC(N3CCN(C)CC3)c2c1. References: Knight J A, etal. Pharmacological analysis of the novel, rapid, and potent...
| Keywords: | Metitepine |
| Application: | 5-HT2 / 5-HT1 antagonist |
| CAS | 19728-88-2 |
| MW: | 472.62 D |
From 77.00€
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Methiothepin (maleate)
Item number: Cay23138-25
Methiothepin is a non-selective antagonist of the serotonin (5-HT) receptor. It is a potent antagonist of 5-HT1A and 5-HT1B (IC50 = 16 nM and Ki = 0.2 nM, respectively) as well as 5-HT2A, 5-HT2B, and 5-HT2C receptors (Kis = 3.16, 2.08, and 4.46 nM, respectively). Methiothepin binds to 5-HT5A, 5-HT5B, 5-HT6, and...
| Keywords: | Metitepine, 1-[10,11-dihydro-8-(methylthio)dibenzo[b,f]thiepin-10-yl]-4-methyl-piperazine, (2Z)-butenedioate |
| Application: | 5-HT2 / 5-HT1 antagonist |
| CAS | 19728-88-2 |
| MW: | 472.6 D |
From 44.00€
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