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GNE-781
Item number: TGM-T15405-100mg
Description: GNE-781 is a highly potent and selective inhibitor of CBP (IC50: 0.94 nM in TR-FRET assay). GNE-781 also inhibits BRET and BRD4(1) (IC50s: 6.2 nM and 5100 nM, respectively). Target: Epigenetic Reader Domain. Smiles: CNC(=O)N1CCc2c(C1)c(nn2C1CCOCC1)N1CCCc2cc(-c3cnn(C)c3)c(cc12)C(F)F. References: Romero...
| Application: | CBP / p300 inhibitor |
| CAS | 1936422-33-1 |
| MW: | 525.59 D |
From 168.00€
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GNE-781
Item number: Cay36450-10
GNE-781 is an inhibitor of CREB-binding protein (CBP) and histone acetyltransferase p300 (IC50s = 0.94 and 1.2 nM, respectively). It is selective for CBP and p300 over bromodomain-containing protein 4 (BRD4) bromodomain 1, BRD4 bromodomain 2, and bromodomain and PHD finger-containing 1 (BRPF1, IC50s = 5.1, 12, and...
| Keywords: | 3-[7-(difluoromethyl)-3,4-dihydro-6-(1-methyl-1H-pyrazol-4-yl)-1(2H)-quinolinyl]-1,4,6,7-tetrahydro-N-methyl-1-(tetrahydro... |
| Application: | CBP / p300 inhibitor |
| CAS | 1936422-33-1 |
| MW: | 525.6 D |
From 504.00€
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