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AM251
AM251

Item number: Cay71670-10

AM251 is a cannabinoid 1 (CB1) receptor 1 antagonist. It binds to CB1 receptors in rat forebrain membrane preparations (Ki = 7.5 nM) and is selective over CB2 receptors in mouse spleen preparations (Ki = 2,290 nM) in radioligand binding assays. AM251 inhibits GTPgammaS binding induced by the CB receptor agonist CP...
Keywords: 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide
Application: SR 141716A analog
CAS 183232-66-8
MW: 555.2 D
From 66.00€ *
Review
AM251
AM251

Item number: LKT-A480000.5

CB1 receptor antagonist/ inverse agonist.
Keywords: AM-251, AM 251, 1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide
Application: SR 141716A analog
CAS 183232-66-8
MW: 555.24 D
From 104.00€ *
Review