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Rupatadine Fumarate
Rupatadine Fumarate

Item number: TGM-T6242-100mg

Description: Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM. Target: Autophagy, PAFR, Histamine Receptor. Smiles: OC(=O)\C=C\C(O)=O.Cc1cncc(CN2CC\C(CC2)=C2/c3ccc(Cl)cc3CCc3cccnc23)c1. References: Merlos M, et al. J Pharmacol Exp Ther, 1997, 280(1),...
Keywords: Alergoliber, Rinialer, Rupafin
Application: Targets histamine receptor H1 (HRH1)
CAS 182349-12-8
MW: 532.03 D
From 33.00€ *
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Rupatadine (fumarate)
Rupatadine (fumarate)

Item number: Cay29478-100

Rupatadine is an antagonist of histamine H1 and platelet-activating factor (PAF) receptors. It binds to rabbit platelet membranes and guinea pig cerebellum membranes with apparent Ki values of 0.55 and 0.1 µM, respectively, in radioligand binding assays. It inhibits contraction of isolated guinea pig ileum induced...
Keywords: 8-chloro-6,11-dihydro-11-[1-[(5-methyl-3-pyridinyl)methyl]-4-piperidinylidene]-5H-benzo[5,6]cyclohepta[1,2-b]pyridine,...
Application: Histamine receptor H1 antagonist, platelet activating factor (PAF) antagonist
CAS 182349-12-8
MW: 532 D
From 209.00€ *
Review