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Conivaptan hydrochloride
Conivaptan hydrochloride

Item number: TGM-T6453-100mg

Description: Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic. Target: Vasopressin Receptor. Smiles: Cl.Cc1nc-2c(CCN(C(=O)c3ccc(NC(=O)c4ccccc4-c4ccccc4)cc3)c3ccccc-23)[nH]1. References: Wada K, et al....
Keywords: Conivaptan HCl, YM 087, Vaprisol
Application: Targets arginine vasopressin receptor 1A (AVPR1A)
CAS 168626-94-6
MW: 535.04 D
From 38.00€ *
Review
Conivaptan (hydrochloride)
Conivaptan (hydrochloride)

Item number: Cay23728-5

Conivaptan is an antagonist of the arginine vasopressin (AVP) receptors V1A and V2 (Kis = 0.48 and 3.04 nM for rat liver V1A and kidney V2, respectively). It also competitively inhibits oxytocin binding to rat uterine oxytocin receptors (Ki = 44 nM) but has no effect on AVP binding to anterior pituitary V1B...
Keywords: YM-087, N-[4-[(4,5-dihydro-2-methylimidazo[4,5-d][1]benzazepin-6(1H)-yl)carbonyl]phenyl]-[1,1'-biphenyl]-2-carboxamide,...
Application: Vasopressin receptor antagonist
CAS 168626-94-6
MW: 535 D
From 94.00€ *
Review