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Rizatriptan benzoate
Item number: TGM-T1512-100mg
Description: Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine headaches. Target: 5-HT Receptor. Smiles: c1cccc(c1)C(=O)O.[nH]1cc(c2cc(ccc12)Cn1ncnc1)CCN(C)C. References: Williamson DJ, et al. Br J...
| Keywords: | MK-462 Benzoate |
| Application: | Targets 5-hydroxytryptamine receptor 1 (HTR1) |
| CAS | 145202-66-0 |
| MW: | 391.47 D |
From 41.00€
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Rizatriptan (benzoate salt)
Item number: Cay16475-10
Rizatriptan is an agonist of the serotonin (5-HT) receptor subtypes 5-HT1B and 5-HT1D (Kis = 4.3 and 10.1 nM, respectively). It is selective for 5-HT1B and 5-HT1D receptors over 5-HT1A receptors (Ki = 140 nM). Rizatriptan induces vasoconstriction in isolated human middle meningeal arteries (EC50 = 90 nM). In vivo,...
| Keywords: | MK-462, N,N-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indole-3-ethanamine, monobenzoate |
| Application: | 5-HT1B / 5-HT1D agonist |
| CAS | 145202-66-0 |
| MW: | 391.5 D |
From 44.00€
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