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CPI-169 racemate
Item number: TGM-T6809-100mg
Description: CPI-169 racemate (CPI 169) is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively. Target: Epigenetic Reader Domain, Histone Methyltransferase. Smiles: CCS(=O)(=O)N1CCC(CC1)C(C)n1c(C)c(C(=O)NCc2c(OC)cc(C)[nH]c2=O)c2ccccc12....
| Keywords: | CPI-169, CPI 169, CPI169 |
| Application: | EZH2 inhibitor |
| CAS | 1450655-76-1 |
| MW: | 528.66 D |
From 53.00€
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CPI-169
Item number: Cay18299-1
The lysine methyltransferase EZH2 (KMT6), part of the polycomb repressive complex 2, catalyzes trimethylation of lysine 27 on histone H3 (H3K27me3) and is involved in proliferation and aggressive cell growth associated with neoplastic cells. CPI-169 is a selective EZH2 inhibitor with IC50 values of 0.24, 0.51, and...
| Keywords: | N-[(1,2-dihydro-4-methoxy-6-methyl-2-oxo-3-pyridinyl)methyl]-1-[1-[1-(ethylsulfonyl)-4-piperidinyl]ethyl]-2-methyl-1H-indo... |
| Application: | EZH2 inhibitor |
| CAS | 1450655-76-1 |
| MW: | 528.7 D |
From 94.00€
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