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Telaglenastat
Telaglenastat

Item number: TGM-T6797-100mg

Description: Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC. Target: Autophagy, transporter, Glutaminase. Smiles: FC(F)(F)Oc1cccc(CC(=O)Nc2ccc(CCCCc3nnc(NC(=O)Cc4ccccn4)s3)nn2)c1. References: Gross MI, et al....
Keywords: CB 839, CB839, CB-839
Application: Targets glutaminase [EC:3.5.1.2] (glsA, GLS)
CAS 1439399-58-2
MW: 571.57 D
From 33.00€ *
Review
CB-839
CB-839

Item number: Cay22038-5

CB-839 is an orally bioavailable noncompetitive inhibitor of the glutaminase 1 (GLS1) splice variants, kidney-type (KGA) and glutaminase C (GAC), which convert glutamine into glutamate. CB-839 inhibits human recombinant GAC with IC50 values of less than 50 nM, varying based on the length of preincubation. It...
Keywords: GLS1 Inhibitor III,...
Application: Glutaminase inhibitor
CAS 1439399-58-2
MW: 571.6 D
From 77.00€ *
Review