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Entacapone
Item number: Cay14153-10
Entacapone is a reversible catechol O-methyltransferase (COMT) inhibitor (IC50s = 10, 10, 20, and 160 nM for rat duodenum, brain, erythrocyte, and liver COMT, respectively). It is selective for COMT over monoamine oxidase A (MAO-A) and MAO-B and phenolsulphotransferase M (PST-M) and PST-P (IC50s = >50 µM)....
| Keywords: | OR-611, 2-cyano-3-(3,4-dihydroxy-5-nitrophenyl)-N,N-diethyl-2E-propenamide |
| Application: | COMT inhibitor |
| CAS | 130929-57-6 |
| MW: | 305.3 D |
From 47.00€
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Entacapone
Item number: AG-CR1-3708-M005
Potent FTO (fat mass and obesity-associated gene) inhibitor for in vivo studies. FTO belongs to the Fe2+ and alpha-ketoglutarate (alpha-KG)-dependent oxygenase family. It demethylates N6-adenosine-modified (m6A) sites and N6,2'-O-dimethyladenosine-modified (m6Am) sites of mRNA. With its demethylase activity, FTO...
| Keywords: | OR-611, (E)-2-Cyano-3-(3,4-dihydroxy-5-nitrophenyl)-N,N-diethylacrylamide |
| Application: | Potent FTO inhibitor (in vivo) |
| CAS | 130929-57-6 |
| MW: | 305.3 D |
From 33.00€
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Entacapone
Item number: TGM-T2216-100mg
Description: Entacapone (OR-611) is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT). Target: Transferase. Smiles: CCN(CC)C(=O)C(=C/c1cc(O)c(O)c(c1)[N+]([O-])=O)\C#N. References: De Santi C, et al. Eur J Clin Pharmacol, 1998, 54(3), 215-219.
| Keywords: | OR-611 |
| Application: | Targets catechol O-methyltransferase [EC:2.1.1.6] (COMT) |
| CAS | 130929-57-6 |
| MW: | 305.29 D |
From 31.00€
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