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Zamifenacin fumarate
Zamifenacin fumarate

Item number: TGM-T13385-100mg

Description: Zamifenacin fumarate (UK-76654 fumarate) is a potent, gut-selective antagonist of the muscarinic M3 receptor. Target: AChR. Smiles: OC(=O)\C=C\C(O)=O.C(Cc1ccc2OCOc2c1)N1CCC[C@H](C1)OC(c1ccccc1)c1ccccc1. References: Houghton LA, et al. Zamifenacin (UK-76, 654) a potent gut M3 selective muscarinic...
Keywords: UK-76654 fumarate
Application: Muscarinic M3 receptor antagonist
CAS 127308-98-9
MW: 531.6 D
From 34.00€ *
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Zamifenacin (fumarate)
Zamifenacin (fumarate)

Item number: Cay32848-1

Zamifenacin is an antagonist of M3 muscarinic acetylcholine receptors (Ki = 10 nM for the human receptor). It is selective for M3 over M1, M2, M4, and M5 receptors in radioligand binding assays using cells expressing recombinant human receptors (Kis = 55, 153, 68, and 34 nM, respectively). Zamifenacin inhibits...
Keywords: UK 76654, (3R)-1-[2-(1,3-benzodioxol-5-yl)ethyl]-3-(diphenylmethoxy)-piperidine, (2E)-2-butenedioate
Application: Muscarinic M3 receptor antagonist
CAS 127308-98-9
MW: 531.6 D
From 43.00€ *
Review