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SR8278
Item number: TGM-T7837-10mg
Description: SR8278 is an REV-ERBalpha antagonist(EC50 = 0.47 µM), blocking activation of the receptor by the synthetic agonist GSK 4112. Target: Others. Smiles: CCOC(=O)C1Cc2ccccc2CN1C(=O)c1ccc(SC)s1. References: Kojetin D , Wang Y , Kamenecka T M , et al. Identification of SR8278, a Synthetic Antagonist of the...
| Application: | NR1D1 antagonist |
| CAS | 1254944-66-5 |
| MW: | 361.48 D |
From 52.00€
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SR8278
Item number: Cay17000-1
REV-ERBalpha is a nuclear receptor and transcription repressor that coordinates circadian rhythm and metabolic pathways in a heme-dependent manner. SR8278 is an antagonist of REV-ERBalpha (EC50 = 0.47 µM), blocking activation of the receptor by the synthetic agonist GSK 4112 (Cay-11931). Moreover, SR8278 stimulates...
| Keywords: | 1,2,3,4-tetrahydro-2-[[5-(methylthio)-2-thienyl]carbonyl]-3-isoquinolinecarboxylic acid, ethyl ester |
| Application: | NR1D1 antagonist |
| CAS | 1254944-66-5 |
| MW: | 361.5 D |
From 61.00€
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