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SB-277011 dihydrochloride
SB-277011 dihydrochloride

Item number: TGM-T12861L-10mg

Description: SB-277011 dihydrochloride is a potent, selective, orally bioavailable and brain penetrate antagonist of dopamine D3 receptor(pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively). Target: Dopamine Receptor. Smiles:...
Keywords: SB-277011A dihydrochloride
Application: DRD3 antagonist
CAS 1226917-67-4
MW: 511.49 D
From 108.00€ *
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SB 277011A (hydrochloride)
SB 277011A (hydrochloride)

Item number: Cay11982-25

SB 277011A is an antagonist of the dopamine D3 receptor (pKi = 8.0) that is at least 100-fold selective for D3 over other monoamine receptors (pKis = 6.0, 5.0, and 2, 5-HT1D and 5-HT1B respectively). It has high oral bioavailability and enters the central nervous system of the rat. SB 277011A has been shown to have...
Keywords: N-[trans-4-[2-(6-cyano-3,4-dihydro-2(1H)-isoquinolinyl)ethyl]cyclohexyl]-4-quinolinecarboxamide, dihydrochloride
Application: DRD3 antagonist
CAS 1226917-67-4
MW: 511.5 D
From 60.00€ *
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