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Nav1.7 Blocker 52
Item number: Cay34477-5
Nav1.7 blocker 52 is an inhibitor of voltage-gated sodium channel 1.7 (Nav1.7, IC50 = 0.17 µM). It is selective for Nav1.7 over human-ether-a-go-go (hERG), also known as Kv11.1, Nav1.5, and Nav1.8 (IC50s = >10, 1.1, and 2.2 µM, respectively) but does inhibit Nav1.3 and Nav1.4 (IC50s = 0.3 and 0.4 µM, respectively)....
| Keywords: | TC-N 1752, Voltage-gated Sodium Channel 1.7,... |
| Application: | Nav1.7 inhibitor |
| CAS | 1211866-85-1 |
| MW: | 516.5 D |
From 163.00€
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TC-N 1752
Item number: TGM-T23439-100mg
Description: TC-N 1752 is an orally active inhibitor of Nav1.7 channel with IC50 of 0.17 µM. TC-N 1752 shows analgesic activities. Target: Sodium Channel. Smiles: CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1C. References: Lin Z, et, al. Biophysical and Pharmacological Characterization of Nav1.9...
| CAS | 1211866-85-1 |
| MW: | 516.52 D |
From 50.00€
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