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Item number: Cay35464-5

Aticaprant is a kappa-opioid receptor (KOR) antagonist (Ki = 0.807 nM). It is selective for KOR over the µ- and delta-opioid receptors (Kis = 24 and 155 nM, respectively). Aticaprant reverses U-69593-induced decreases in nocifensive behavior in the formalin test in rats (ED50 = 0.4 mg/kg). It also reverses...

Keywords:	CERC-501, JNJ-67953964, LY2456302, 4-[4-[[(2S)-2-(3,5-dimethylphenyl)-1-pyrrolidinyl]methyl]phenoxy]-3-fluoro-benzamide
Application:	Kappa-opioid receptor antagonist
CAS	1174130-61-0
MW:	418.5 D

From 145.00€ *

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Aticaprant

Item number: TGM-TQ0082-100mg

Description: Aticaprant (LY-2456302) (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM). Target: Opioid Receptor. Smiles: Cc1cc(C)cc(c1)[C@@H]1CCCN1Cc1ccc(Oc2ccc(cc2F)C(N)=O)cc1. References: Rorick-Kehn LM, et al. LY2456302 is a novel, potent, orally-bioavailable...

Keywords:	LY-2456302, CERC-501
Application:	Targets kappa-type opioid receptor (OPRK1)
CAS	1174130-61-0
MW:	418.5 D

From 34.00€ *

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