2 products were found matching "1164500-72-4"!

No results were found for the filter!
ML 145
ML 145

Item number: TGM-T12074-2mg

Description: ML 145 is a selective antagonist of GPR35/CXCR8 (IC50/EC50 of 20.1 nM). Target: Others. Smiles: C\C(\C=C1/SC(=S)N(CCCC(=O)Nc2ccc(C(O)=O)c(O)c2)C1=O)=C/c1ccccc1. References: Heynen-Genel S, et al. Selective GPR35 Antagonists - Probes 1 & 2. National Center for Biotechnology Information (US), 2010-2010...
Application: GPR35 antagonist
CAS 1164500-72-4
MW: 482.57 D
91.00€ *
Review
ML-145
ML-145

Item number: Cay33534-1

ML-145 is an antagonist of G protein-coupled receptor 35 (GPR35). It inhibits beta-arrestin recruitment induced by the GPR35 agonists zaprinast (Cay-10010421), cromolyn (Cay-21379), and pamoic acid (Cay-13946) in HEK293 cells expressing the human receptor (EC50s = 26, 22, and 8.3 nM, respectively). ML-145 inhibits...
Keywords: 2-hydroxy-4-[[4-[(5Z)-5-[(2E)-2-methyl-3-phenyl-2-propen-1-ylidene]-4-oxo-2-thioxo-3-thiazolidinyl]-1-oxobutyl]amino]-benz...
Application: GPR35 antagonist
CAS 1164500-72-4
MW: 482.6 D
From 85.00€ *
Review