2 products were found matching "1125758-85-1"!
No results were found for the filter!
A-804598
Item number: TGM-T3639-100mg
Description: A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat, 9 nM, mouse, 11 nM, human). Target: P2X Receptor. Smiles: C[C@H](N(C(=N)NC#N)c1cccc2ncccc12)c1ccccc1. References: Donnelly-Roberts DL, et al. Neuropharmacology. 2009 Jan,56(1):223-9.
| Keywords: | A 804598 |
| Application: | P2X7 antagonist |
| CAS | 1125758-85-1 |
| MW: | 315.37 D |
From 25.00€
*
A-804598
Item number: Cay20060-10
A-804598 is a potent and selective competitive antagonist of the purinergic P2X7 receptor, a ligand-gated ion channel, with IC50 values of 9.9 and 10.9 nM in 132N1 cells transfected with the rat or mouse receptor, respectively. It inhibits IL-1beta release in human THP-1 cells stimulated with LPS and IFN-gamma (IC50...
| Keywords: | N-cyano-N''-[(1S)-1-phenylethyl]-N'-5-quinolinyl-guanidine |
| Application: | P2X7 antagonist |
| CAS | 1125758-85-1 |
| MW: | 315.4 D |
From 128.00€
*
