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LP-211
Item number: TGM-T5387-100mg
Description: LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor. Target: 5-HT Receptor, Dopamine Receptor. Smiles: C(CCCCC(NCC1=CC=C(C#N)C=C1)=O)N2CCN(C3=C(C=CC=C3)C4=CC=CC=C4)CC2. References: Leopoldo M, et al. Structural...
| Application: | 5-HT7 agonist |
| CAS | 1052147-86-0 |
| MW: | 466.62 D |
From 40.00€
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LP-211
Item number: Cay29659-10
LP-211 is an agonist of the serotonin (5-HT) receptor subtype 5-HT7 (Ki = 0.58 nM). It is selective for 5-HT7 over 5-HT1A and dopamine D2 receptors (Kis = 188 and 142 nM, respectively). It induces relaxation of isolated guinea pig ileum precontracted by substance P (Cay-24035, EC50 = 0.6 µM). LP-211 (100 nM)...
| Keywords: | 4-[1,1'-biphenyl]-2-yl-N-[(4-cyanophenyl)methyl]-1-piperazinehexanamide |
| Application: | 5-HT7 agonist |
| CAS | 1052147-86-0 |
| MW: | 466.6 D |
From 44.00€
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