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CARM1-IN-1
CARM1-IN-1

Item number: TGM-T10682L-100mg

Description: CARM1-IN-1 (CARM1-IN-7G) is a selective inhibitor of CARM1 with IC50 of 8.6 µM. CARM1-IN-1 shows weak activity against PRMT1 and SET7 with IC50 > 600 µM. Target: Histone Methyltransferase. Smiles: Oc1ccc(\C=C2/CN(Cc3ccccc3)C\C(=C/c3ccc(O)c(Br)c3)C2=O)cc1Br. References: Cheng D, et al. Novel...
Keywords: CARM1-IN-7G
CAS 1020399-49-8
MW: 555.26 D
From 31.00€ *
Review
PRMT4/CARM1 Inhibitor
PRMT4/CARM1 Inhibitor

Item number: Cay11033-1

PRMT4/CARM1 Inhibitor selectively blocks the activity of PRMT4/CARM1 with an IC50 value of 7.1 µM. It displays very low affinity towards PRMT1 and SET7 with IC50 values of 63 and 943 µM, respectively. In human prostate cancer LNCaP cells, this compound reduced the prostate-specific antigen promoter activity at 8-10...
Keywords: Protein Arginine Methyltransferase 4/Coactivator-Associated Arginine Methyltransferase 1 Inhibitor,...
CAS 1020399-49-8
MW: 555.3 D
From 111.00€ *
Review