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Item number: TGM-T15786-10mg

Description: LPA2 antagonist 1 is an LPA2 antagonist (IC50: 17 nM). Target: Hydroxylase. Smiles: C[C@@H](CN1CCN(CC1)S(=O)(=O)c1ccc(Cl)c(Cl)c1)Nc1ncnc2c(C)csc12. References: Beck HP, et al. Discovery of potent LPA2 (EDG4) antagonists as potential anticancer agents. Bioorg Med Chem Lett. 2008 Feb 1,18(3):1037-41.

Application:	LPAR2 antagonist
CAS	1017606-66-4
MW:	500.46 D

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LPA2 Antagonist 1

Item number: Cay22051-1

LPA2 antagonist 1 is an antagonist of lysophosphatidic acid receptor 2 (LPA2, IC50 = 17 nM). It is selective for LPA2 over LPA1 and LPA3 (IC50s = >50 µM). LPA2 antagonist 1 inhibits HGF-induced phosphorylation of ERK and proliferation of HCT116 colon cancer cells in a concentration-dependent manner.Formal Name:...

Keywords:	LPA2-IN-1, N-[(1S)-2-[4-[(3,4-dichlorophenyl)sulfonyl]-1-piperazinyl]-1-methylethyl]-7-methyl-thieno[3,2-d]pyrimidin-4-amine
Application:	LPAR2 antagonist
CAS	1017606-66-4
MW:	500.5 D

From 323.00€ *

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