(S)-Enitociclib

Item number	Size	Delivery time	Price
TGM-T70388-1mg	1 mg	7 - 10 business days*	516.00€
TGM-T70388-2mg	2 mg	7 - 10 business days*	752.00€
TGM-T70388-5mg	5 mg	7 - 10 business days*	1,170.00€
TGM-T70388-10mg	10 mg	7 - 10 business days*	1,430.00€
TGM-T70388-25mg	25 mg	7 - 10 business days*	1,921.00€
TGM-T70388-50mg	50 mg	7 - 10 business days*	2,382.00€

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Description: (S)-Enitociclib (VIP152) is a selective CDK9 inhibitor that induces complete... more

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Product information "(S)-Enitociclib"

Description: (S)-Enitociclib (VIP152) is a selective CDK9 inhibitor that induces complete regression of MYC+ lymphomas by inhibiting RNA polymerase II-mediated transcription of anti-apoptotic and pro-survival proteins. Target: CDK. Smiles: COC1=C(C2=C(F)C=NC(NC3=CC(C[S@@](C)(=N)=O)=CC=N3)=C2)C=CC(F)=C1. References: Lücking U,et al. Changing for the Better: Discovery of the Highly Potent and Selective CDK9 Inhibitor VIP152 Suitable for Once Weekly Intravenous Dosing for the Treatment of Cancer. J Med Chem. 2021 Aug 12,64(15):11651-11674.

Keywords:	VIP152
Supplier:	TargetMol
Supplier-Nr:	T70388

Properties

Application:	Targets cyclin-dependent kinase 9 [EC:2.7.11.22 2.7.11.23] (CDK9)
MW:	404.43 D
Formula:	C19H18F2N4O2S
Format:	32160405

Database Information

CAS :	1610408-97-3\| Matching products
KEGG ID :	K02211 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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