Repotrectinib

Item number	Size	Delivery time	Price
TGM-T4071-1mg	1 mg	7 - 10 business days*	45.00€
TGM-T4071-2mg	2 mg	7 - 10 business days*	63.00€
TGM-T4071-5mg	5 mg	7 - 10 business days*	97.00€
TGM-T4071-1mL	1 ml	7 - 10 business days*	102.00€
TGM-T4071-10mg	10 mg	7 - 10 business days*	172.00€
TGM-T4071-25mg	25 mg	7 - 10 business days*	311.00€
TGM-T4071-50mg	50 mg	7 - 10 business days*	497.00€
TGM-T4071-100mg	100 mg	7 - 10 business days*	724.00€

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Description: Repotrectinib (TPX-0005) is a potent ALK/ROS1/TRK inhibitor, with IC50 values of... more

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Product information "Repotrectinib"

Description: Repotrectinib (TPX-0005) is a potent ALK/ROS1/TRK inhibitor, with IC50 values of 1.01 nM for WT ALK, 5.3 nM for SRC, 1.08 nM for ALK L1196M, and 1.26 nM for ALK G1202R. Target: ALK, ROS, ROS Kinase, Src, Trk receptor. Smiles: C[C@H]1CNC(=O)c2cnn3ccc(N[C@H](C)c4cc(F)ccc4O1)nc23. References: Dayong Zhai, et al. Abstract 2132: The novel, rationally-designed, ALK/SRC inhibitor TPX-0005 overcomes multiple acquired resistance mechanisms to current ALK inhibitors. Cancer Research. July 2016

Keywords:	TPX-0005, TPX0005, TPX 0005
Supplier:	TargetMol
Supplier-Nr:	T4071

Properties

Application:	Targets proto-oncogene tyrosine-protein kinase ROS [EC:2.7.10.1] (ROS1)
MW:	355.37 D
Formula:	C18H18FN5O2
Format:	32160405

Database Information

CAS :	1802220-02-5\| Matching products
KEGG ID :	K03176 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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