Preladenant
If you have any questions, please use our Contact Form.
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A... more
Product information "Preladenant"
Description: Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine receptors. Target: Adenosine Receptor. Smiles: COCCOc1ccc(cc1)N1CCN(CCn2ncc3c2nc(N)n2nc(nc32)-c2ccco2)CC1. References: Hodgson RA, et al. Characterization of the potent and highly selective A2A receptor antagonists preladenant and SCH 412348 [7-[2-[4-2,4-difluorophenyl]-1-piperazinyl]ethyl]-2-(2-furanyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine] in rodent models of movement disorders and depression. J Pharmacol Exp Ther. 2009 Jul,330(1):294-303.
| Keywords: | SCH-420814 |
| Supplier: | TargetMol |
| Supplier-Nr: | T4290 |
Properties
| Application: | Targets adenosine receptor A2a (ADORA2A, ADOR) |
| MW: | 503.56 D |
| Formula: | C25H29N9O3 |
Database Information
| CAS : | 377727-87-2| Matching products |
| KEGG ID : | K04266 | Matching products |
Handling & Safety
| Storage: | +4°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Danger |
| GHS Hazard Pictograms: |
|
| H Phrases: | H319, H361, H372, H410 |
| P Phrases: | P201, P202, P260, P264, P270, P273, P280, P314, P391, P305+P351+P338, P308+P313, P337+P313, P405, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
You will get a certificate here
Viewed