PF-5190457
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi:... more
Product information "PF-5190457"
Description: PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36). Target: GHSR. Smiles: Cc1cn2cc(CC(=O)N3CCC4(CN(C4)[C@@H]4CCc5cc(ccc45)-c4cc(C)ncn4)CC3)nc2s1. References: Bhattacharya SK, et al. Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor Inverse Agonist Clinical Candidate. ACS Med Chem Lett. 2014 Feb 24,5(5):474-9.
| Keywords: | PF-05190457 |
| Supplier: | TargetMol |
| Supplier-Nr: | T16508 |
Properties
| Application: | GHS-R inverse agonist |
| MW: | 512.67 D |
| Formula: | C29H32N6OS |
Database Information
| CAS : | 1334782-79-4| Matching products |
| KEGG ID : | K04284 | Matching products |
Handling & Safety
| Storage: | +4°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H315, H319 |
| P Phrases: | P264, P280, P302+352, P305+351+338, P321, P332+313, P337+313, P362+364 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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