PF-4981517

Item number	Size	Manual	Delivery time	Price
TGM-T21548-1mg	1 mg	-	7 - 10 business days*	41.00€
TGM-T21548-5mg	5 mg	-	7 - 10 business days*	95.00€
TGM-T21548-10mg	10 mg	-	7 - 10 business days*	151.00€
TGM-T21548-25mg	25 mg	-	7 - 10 business days*	305.00€
TGM-T21548-50mg	50 mg	-	7 - 10 business days*	-

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Description: PF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of... more

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Product information "PF-4981517"

Description: PF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4). The IC 50 values for CYP3A activity are 0.03 µM,17 µM, and 71 µM for CYP3A4, CYP3A5, and CYP3A7, respectively. PF-4981517 is able to be used to distinguish the contributions of CYP3A4 versus CYP3A5 on drug Metabolism. Target: P450. Smiles: Cc1ccc(cc1)-c1c(cnn1C)-c1nn(C)c2ncnc(N3CC[C@@H](C3)N3CCCCC3)c12. References: Robert L Walsky, et al. Selective mechanism-based inactivation of CYP3A4 by CYP3cide (PF-04981517) and its utility as an in vitro tool for delineating the relative roles of CYP3A4 versus CYP3A5 in the metabolism of drugs. Drug Metab Dispos. 2012 Sep,40(9)

Keywords:	CYP3cide
Supplier:	TargetMol
Supplier-Nr:	T21548

Properties

Application:	CYP3A4 inhibitor
MW:	456.59 D
Formula:	C26H32N8

Database Information

CAS :	1390637-82-7\| Matching products
KEGG ID :	K17689 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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